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4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-[(3R,4R)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
2-[(2-chlorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4-methoxyphenyl)propanamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-4-(2-oxopyrrolidin-1-yl)benzamide
5-chloro-3-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-[3-(4-fluorophenyl)phenyl]piperidin-4-amine
4-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
6,6-dimethyl-1-phenyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(3,4-dichlorophenyl)-4-(6-phenylpyridazin-3-yl)morpholine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
6-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-9H-purin-2-amine
({4-cyclopropyl-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-chloro-N,1-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}piperidin-2-one
1-(3-chlorophenyl)-4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-2-one
(2-methoxyethyl)(methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(1-ethylpiperidine-3-carbonyl)piperidine
1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-phenylazepane
5-[1-(butan-2-yl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(quinolin-6-ylmethyl)-1-benzofuran-2-carboxamide
4-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
1-(2-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}ethyl)pyrrolidin-2-one
{4-[(6-ethoxyquinolin-2-yl)methyl]morpholin-2-yl}methanamine
4-(1H-imidazol-2-yl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
2-[4-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
2-(2-methoxyethyl)-4-[(2-propoxynaphthalen-1-yl)methyl]morpholine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
(2R)-N-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-2-(hydroxymethyl)pyrrolidine-1-carboxamide
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
2-(1-benzothiophen-7-yl)-5-methylpyrimidin-4-amine
1-(3-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
2-chloro-4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]oxane-2-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-methyl-N-(1-methylpyrrolidin-3-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4,6-dimethoxy-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-chloro-3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
(benzylsulfamoyl)[2-(1H-imidazol-1-yl)-1-phenylethyl]amine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
(4aR,8aS)-1-butyl-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-({3-[2-(hydroxymethyl)piperidin-1-yl]propyl}amino)pyrimidine-5-carboxylic acid
4-cyano-1-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-pyrrole-2-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
9-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one