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ethyl 4-({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)piperidine-1-carboxylate
N-ethyl-3-(1H-indol-3-yl)-N-(oxan-4-yl)propanamide
3-phenyl-1-[1-(quinoline-8-carbonyl)piperidin-3-yl]propan-1-one
N-(4,5-dihydro-1,3-thiazol-2-yl)-2-{5-[(N-methylacetamido)methyl]-1,2,3,6-tetrahydropyridin-1-yl}propanamide
3-[(dimethylamino)methyl]-1-[(2-phenylphenyl)methyl]piperidin-3-ol
3-(1-{[1-(4-methylphenyl)propan-2-yl]amino}ethyl)adamantan-1-ol
4-(2H-1,3-benzodioxol-5-yloxy)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
1-methyl-N-[3-(phenylsulfanyl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(3R,4S)-1-(3-chlorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-2-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyrimidine
N-methyl-4-{1-[(2-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}-1,3-thiazol-2-amine
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2,3-dimethylquinoxaline-6-carboxamide
8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-4-amino-1-(1-benzylpiperidin-4-yl)-N,N-diethylpyrrolidine-2-carboxamide
ethyl 1-(3-methylbutyl)-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[(4aR,7aS)-4-[(2-chlorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-phenylethane-1,2-dione
4-(1-methyl-1H-imidazol-2-yl)-N-(4-phenoxyphenyl)piperidine-1-carboxamide
2-methoxyethyl 3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-hydroxy-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
6-(cyclopentylmethyl)-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
(2S)-3-(4-hydroxyphenyl)-2-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamido]propanamide
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
6-methyl-2-({2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
2-(4-fluorophenoxymethyl)-4-hydroxy-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-5-carboxamide
N-({5-[4-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[3-(1,3-benzothiazol-2-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-methyl-8-[2-(4-propanoylphenoxy)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-3,4-dihydroquinazolin-4-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(4-methoxy-3-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-amino-2-{4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-(1,3-benzoxazol-2-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-methyl-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2,3,6-tetrahydropyridine
5-(4-methoxyphenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
5,8-dimethyl-2-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)quinolin-4-ol
8-fluoro-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinoline-2-carboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(4-hydroxybutyl)piperidine-3-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(propan-2-yl)pyrimidine-4-carboxamide
(1S,2S)-N2-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-2,3-dihydro-1H-indene-1,2-diamine
2-(4-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}quinolin-4-ol
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
7-(5-chlorothiophen-2-yl)-1,2-dihydroisoquinolin-1-one
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine