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5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-({[1-(4,7-dimethylquinazolin-2-yl)azepan-4-yl]amino}methyl)hepta-1,6-dien-4-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(4-chloro-2-methylphenoxy)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}propan-1-one
1-(2-methoxyphenyl)-3-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(3S,4S)-1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-3,4-diol
2-[(3,4-difluorophenyl)methyl]-N,N-dimethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(5-methyl-1H-indol-3-yl)pyridine-3-carbonitrile
3-[4-(benzenesulfonyl)piperazine-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(3-methoxypropyl)amine
1-methyl-3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-cyclopentyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-5-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
5-[4-(aminomethyl)piperidin-1-yl]-2-(2-phenylethyl)-2,3-dihydropyridazin-3-one
3-(2,3-dihydro-1-benzofuran-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-acetamido-N-(1H-indol-2-ylmethyl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(2R,3R)-3-{[2-(2-methoxyphenyl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
8-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{2-[(2-amino-4-methyl-1,3-benzothiazol-6-yl)formamido]ethyl}pyridine-3-carboxamide
4-{4-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]phenyl}morpholine
3-(4-methyl-1,3-thiazol-5-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
3-{3-[(2-fluorophenyl)formamido]propanamido}hexanoic acid
(2-ethoxy-5-{[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)methanol
2-(dimethyl-1,3-thiazol-5-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
N-[(3R,4R)-1-(2-cyclopentylacetyl)-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
(3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-oxopropyl)urea
4-[(2-ethylphenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(1-methyl-1H-indazol-3-yl)benzamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(4-methylpentanoyl)piperidine-4-carboxamide
2-{2-[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
1-[3-(morpholin-4-yl)piperidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
(3S)-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidine-3-carboxylic acid
3-[methyl({[2-(trifluoromethyl)phenyl]methyl})carbamoyl]benzoic acid
6-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
2-(furan-2-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[1-(2-methylbutyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-{1-oxaspiro[4.4]nonan-3-yl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(1H-pyrazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-methyl-6-(4-{[2-(2-methyl-1H-indol-3-yl)ethyl]amino}piperidin-1-yl)pyrimidin-2-amine
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-4-phenyl-N-(pyridin-2-ylmethyl)benzamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[1-(piperidine-1-carbonyl)piperidin-4-yl]acetamide
3-[(methylsulfanyl)methyl]-5-(5-phenyl-1,2-oxazol-3-yl)-1,2,4-oxadiazole
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]propanamide
N-benzyl-3-(1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperidin-4-yl)-N-methylpropanamide