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[(2S,4R)-4-(dimethylamino)-1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-2-yl]methanol
2-({6-[(E)-2-cyclohexylethenyl]pyridazin-3-yl}(methyl)amino)ethan-1-ol
4-({3-azaspiro[5.5]undecan-9-yl}amino)-1-propylpyrrolidin-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(1R)-2-hydroxy-1-phenylethyl]propanamide
4-ethyl-3-{1-[3-(pyrimidin-2-yloxy)benzoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-N-cycloheptyl-4-(1H-1,2,3,4-tetrazol-1-yl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-{4-[(2-hydroxyethyl)(methyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[2-(2-chlorophenoxy)ethyl]-N-ethyl-1,7-dimethyl-1H-indole-2-carboxamide
5-(2-ethoxyethyl)-3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
methyl 2-{1-[4-(azocan-1-yl)-5-methylthieno[2,3-d]pyrimidin-6-yl]-N-methylformamido}acetate
3-methyl-7-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(4-methyl-1H-pyrazol-3-yl)piperidine
{2-fluoro-5-[6-(pyrrolidin-1-yl)pyridazin-3-yl]phenyl}methanol
5-phenyl-3-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,2-oxazole
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[1-(pyridin-3-yl)propyl]amine
2-[(1-methylpiperidin-3-yl)methyl]-1,2-dihydrophthalazin-1-one
N-[2-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]acetamide
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
1,3-dimethyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1H-pyrazole-4-carboxamide
6-(2-aminoethyl)-N,2-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidin-4-amine
7-(3-hydroxy-4-methoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[1-(furan-3-ylmethyl)-4-[3-(5-methylfuran-2-yl)benzoyl]piperazin-2-yl]ethan-1-ol
3-{2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
5-[1-(2,5-dimethylphenoxy)ethyl]-3-methyl-1H-1,2,4-triazole
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-4-(diphenylmethyl)piperazine
N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-(pyrrolidin-1-ylmethyl)-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-ol
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(thiolan-3-yl)benzamide
2,3,5-trimethyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,4-dihydropyridine-3-carboxamide
N-methyl-2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]acetamide
4-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3,5-dimethyl-1,2-oxazole
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(2-methylpropyl)piperidin-4-yl]methyl}amine
4-{4-[2-(morpholin-4-ylmethyl)phenyl]phenyl}-1,3-thiazol-2-amine
4-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
1-{2-[1-(1-benzofuran-3-carbonyl)piperidin-2-yl]ethyl}-4-methylpiperazine
1-(3-methylphenyl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
7-{[4-(dimethylamino)azepan-1-yl]methyl}-2-ethyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
4-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(2-aminoethyl)-N-methyl-N-(quinoxalin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-[4-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
7-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dimethyl-1H-indole
1-(furan-2-ylmethyl)-4-[(1E)-1-phenylprop-1-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)acetamide
2-cyclopentyl-N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}acetamide
1-[2-(2-ethoxyethoxy)phenyl]-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-methylurea