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(2S,4R)-N-ethyl-4-{[(4-phenylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
3-(2-cyanophenyl)-5-[(oxolan-2-ylmethyl)sulfamoyl]benzoic acid
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
(3S,4R)-1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidine
5-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
6-{[(3R,4S)-4-cyclopropyl-1-(3-methylbut-2-enoyl)pyrrolidin-3-yl]amino}pyrazine-2-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
N-[(3S,4R)-1-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-4-propylpyrrolidin-3-yl]acetamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-indol-1-yl)ethyl]amine
4-[(5-{1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]-3-methylbut-2-en-1-one
6-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carbonitrile
N,5-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(1-phenylcyclopentyl)methyl]propanamide
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
3-{2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-methylcyclohexanamine
N-[2-(2-chloro-6-methylphenoxy)ethyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
1-(1-cyclobutylethyl)-4-(cyclopropylmethyl)-1,4-diazepan-5-one
N-(3-hydroxy-3-phenylpropyl)-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N,1-dimethyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-(3-hydroxybenzoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(3-methoxyphenyl)methyl]piperidine
N-(5-chloro-2-methoxyphenyl)-3-[1-(quinoline-3-carbonyl)piperidin-3-yl]propanamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1,4-diazepan-1-yl}-4,6,7-trimethylquinazoline
(3R)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-ol
2,6-dimethyl-4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]quinoline
N-(2-methoxyethyl)-6-[3-(methoxymethyl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-{2-[2-(trifluoromethoxy)phenyl]pyrimidin-4-yl}piperidin-4-ol
2-{3-[3-(trifluoromethyl)phenoxymethyl]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3S)-4-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidine
2-(2-hydroxyethyl)-9-{[2-(methylsulfanyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[(2-chlorophenyl)methyl]-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)carbamoyl}amino)-2-methyl-N-(2-methylpropyl)benzamide
N-(furan-2-ylmethyl)-5-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
7-(cyclopropylmethyl)-2-(naphthalene-1-carbonyl)-2,7-diazaspiro[4.5]decane
2-{[4-(4-hydroxyphenyl)phenyl]sulfanyl}acetamide
{5-chloro-7-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
(1R,3S)-7-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(2-methoxyphenyl)methyl]propylamine
(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-3,6-dimethylquinoline
1-(2,3-dihydro-1H-inden-4-yl)-3-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
(3R,5R)-5-[4-(4-methoxybenzenesulfonyl)piperazine-1-carbonyl]pyrrolidin-3-ol
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide