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3-(2-methoxybenzoyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-(3-{4-[(2-hydroxy-2-phenylethyl)(methyl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
N-[(3S,4R)-1-(6-cyanopyridin-2-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-(dimethylamino)-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(2-methylphenyl)acetamide
[2-(2,3-dihydro-1H-indol-1-yl)ethyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
3-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
1-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]-6-[1-(methylsulfanyl)propan-2-yl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-amino-6-(1H-pyrrol-2-yl)-4-(2,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
N-[(3S,4R)-4-(4-methylphenyl)-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]acetamide
2-acetyl-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(6-methylpyridazin-3-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N3-{2-[(2-methylquinolin-8-yl)oxy]ethyl}piperidine-1,3-dicarboxamide
N4-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(1S,2S,4R)-1,7,7-trimethyl-4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]bicyclo[2.2.1]heptan-2-ol
(4aR,7aS)-1-cyclopropanecarbonyl-4-(2,6-dimethylpyrimidine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(butylsulfanyl)-N4-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyrimidine-4,6-diamine
7-methyl-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
(1,3-benzothiazol-2-ylmethyl)({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(1H-indol-3-yl)propan-1-one
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(2-methylphenyl)-1,4-diazepane
5-(morpholin-4-ylmethyl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]furan-3-carboxamide
ethyl 4-[(1-{4-[(benzylcarbamoyl)methyl]phenyl}piperidin-4-yl)amino]piperidine-1-carboxylate
4-[(3-{3-methyl-1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]morpholine
8-(1,2,3,4-tetrahydroisoquinolin-7-yl)quinoline
5-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
7-[(4-fluorophenyl)methyl]-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(furan-2-yl)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole
5-{4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-{[6-(dimethylamino)pyridin-3-yl]methyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{4-[(2-cyclohexylpyrimidin-5-yl)methyl]-1,4-oxazepan-6-yl}methanol
1-(2-phenylethyl)-4-[(pyridin-4-ylmethyl)amino]pyrrolidin-2-one
N'-(2,3-dihydro-1H-inden-2-yl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-N'-methylethanediamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxane-4-carboxamide
1-(1,4-dithiepan-6-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1H-pyrazole
5-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]quinoline-4-carboxylic acid
1-ethyl-N-[(2-fluorophenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,5R)-3-[(3E)-4-methylhex-3-en-1-yl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(4-methoxyphenyl)-3-methyl-4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazin-2-one
(3S,4S)-1-(3-aminobenzoyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
2-({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(propan-2-yl)amino)ethan-1-ol
2-(dimethyl-1,3-thiazol-4-yl)-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
(3R,4R)-4-(azepan-1-yl)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-ol
N-(3-chloro-4-fluorophenyl)-3-[3-(dimethylamino)pyrrolidin-1-yl]-3-oxopropanamide
6-methyl-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxylic acid
9-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one