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4-[5-(2,3-dihydro-1H-isoindol-2-ylmethyl)-1,2,4-oxadiazol-3-yl]benzoic acid
3-chloro-N-(1H-imidazol-2-ylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-(4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-cyclopentyl-N-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-cyclopropyl-1-phenyl-1H-1,2,4-triazole
2-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-6-(morpholine-4-carbonyl)pyrazin-2-amine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
5-{4-[2-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[(4-fluorophenyl)methyl]-4-(pyridin-2-ylmethyl)morpholine
3-(2-phenoxyethyl)-1-(1,3-thiazol-2-yl)piperidine-3-carboxylic acid
4-[(2S)-1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}pyrrolidine-2-carbonyl]morpholine
2-{4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
3-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}piperidin-3-ol
3-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
1-cyclopentanecarbonyl-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
1-(4-methyl-1,4-diazepane-1-carbonyl)-6-[(2,4,5-trimethoxyphenyl)methyl]-6-azaspiro[2.5]octane
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(cyclopropylmethyl)-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-propyl-1H-pyrazole-4-carboxamide
N-[2-(1H-imidazol-1-yl)propyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-(2-methylphenyl)piperidine
(1R,3S)-3-(2-aminoethoxy)-7-(2,5-dimethylfuran-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N-methyl-N-{2-[2-(quinolin-4-yl)-1H-imidazol-1-yl]ethyl}methanesulfonamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
(3R,4R)-4-(morpholin-4-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-ol
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-(piperidin-1-ylmethyl)piperidin-2-one
8-[(2,5-dimethylphenyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-methyl-2-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
2-(3-chloro-4-fluorobenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
4-{6-azaspiro[2.5]octane-1-carbonyl}-1-(4-methoxyphenyl)piperazin-2-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methyl-3-(morpholin-4-yl)propanamide
1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-ol
5-oxo-1-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxylic acid
3-{4-[(2-phenylazetidin-1-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
4-(2H-1,3-benzodioxol-5-ylmethyl)-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
14-[(benzyloxy)methyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-(piperazine-1-carbonyl)-N-[2-(pyridin-2-yl)ethyl]benzene-1-sulfonamide
2-(3,4,5-trifluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 1-{2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetyl}piperidine-4-carboxylate
N-(cyclopropylmethyl)-N-methyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
methyl 4-oxo-4-(4-{2-[(pyridin-3-ylmethyl)carbamoyl]ethyl}piperidin-1-yl)butanoate
1-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
{4-[(3,5-dichloropyridin-4-yl)methyl]-1,4-oxazepan-6-yl}methanol