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N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-2-phenylpropanamide
2-(oxolan-2-ylmethyl)-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(morpholin-4-yl)ethyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
9-hydroxy-4-oxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1-ethyl-5-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-({methyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)pyridine-3-carboxylic acid
2-[2-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)phenoxy]acetic acid
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(pyridin-3-yl)ethyl]amino}methyl)piperidin-2-one
2-(3-methoxypropyl)-8-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)acetamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethan-1-one
2-(2-methoxyethyl)-9-[2-(methylsulfanyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,3-benzothiazol-6-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-5,6-dimethylpyridine-3-carboxamide
N-[2-(3-chlorophenyl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
methyl({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(pyridin-2-ylmethyl)amine
(1R,7S)-3-tert-butyl-N-methyl-4-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 9-[3-(dimethylamino)propoxy]-7-oxo-3-[4-(1H-pyrazol-1-yl)benzoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(1H-imidazol-2-yl)propyl]benzamide
3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propanamide
2-(2-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)propanamide
2-[2-oxo-4-(5-phenylpentanoyl)piperazin-1-yl]benzonitrile
N-methyl-2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
14-(5-ethylfuran-2-yl)-6-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
methyl({[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
(3R,5R)-N-cyclopropyl-1-(naphthalen-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
1-[6-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
4-[(5-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
(2R)-2-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
methyl 3-chloro-4-{[(oxan-4-yl)carbamoyl]amino}benzoate
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
[2-(azepan-1-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-(2,2-dimethyloxan-4-yl)-2-(thiophen-2-yl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[(6-methylpyridin-2-yl)methyl]piperidin-4-ol
(furan-2-ylmethyl)({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})(thiophen-3-ylmethyl)amine
4,5-dimethyl-6-[4-(trifluoromethyl)piperidin-1-yl]pyrimidine
8-fluoro-3-[1-(1H-pyrazol-1-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{spiro[2.5]octan-1-ylmethyl}-1,3-oxazole-4-carboxamide
4-methyl-5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-(methylsulfanyl)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
5-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylbenzene-1,3-diol
1-{1-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperidin-4-yl}-1,4-diazepan-5-one
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
2-(3-methoxyphenyl)-5-(oxan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[(2-methylphenyl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide