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2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}acetamide
2-{4-[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-imidazol-1-yl}-6-methylpyridine
(1S,4S)-2-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
N-[4-(1H-pyrazol-1-yl)butan-2-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
4-ethyl-3-({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1,2-oxazole
N,N-diethyl-1-[2-(1H-imidazol-2-yl)benzoyl]pyrrolidin-3-amine
methyl 8-(3-methylbut-2-en-1-yl)-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{[(3-methyl-1H-pyrazol-5-yl)methyl](pyridin-2-ylmethyl)amino}butan-1-ol
5-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-2,3-dimethyl-1H-indole
2-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
(2S,4R)-1-[(4-hydroxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(piperidin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-ethylurea
3-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-3,9-diazaspiro[5.5]undecane
N-(1-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-(1-propylcyclopropyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(isoquinoline-1-carbonyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]acetamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-5-methoxy-4-oxo-4H-pyran-2-carboxamide
N-[3-(methylamino)propyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(3-chlorophenyl)methyl]-6-(morpholine-4-carbonyl)-1,3-benzoxazole
N-cyclopropyl-1-(1-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperidin-4-yl)piperidine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-ol
1-[1-ethyl-5-(naphthalen-1-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
N-(furan-2-ylmethyl)-N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}propanamide
7-(cyclobutylmethyl)-2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[3-(phenylsulfanyl)propyl]amine
dimethyl({4-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)amine
[1-(6-aminopyrimidin-4-yl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
3-{5-[2-methyl-2-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-methyl-4-phenylpyridine-3-carboxamide
1-[(2-ethoxyphenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-fluorophenyl)piperazine
4-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2-methylphenol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
{2-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl}bis(propan-2-yl)amine
2-{[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]methyl}-4-methyl-6-(trifluoromethyl)pyrimidine
1-[(4-methylphenyl)methyl]-4-(2,3,6-trifluorobenzoyl)piperazin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
5-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-(furan-2-carbonyl)pyrrolidin-3-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide