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2-(2,3-dihydro-1H-inden-1-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-methyl-5-(2-methylphenyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,4-triazin-3-amine
1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]pentane-1,2-dione
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)pyrimidin-2-amine
4-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
4-methyl-2-{2-oxo-2-[4-(pyridin-4-yloxy)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopropane-1-carboxamide
1-(2,2-dimethyloxane-4-carbonyl)-4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
5-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
5-methyl-4-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)thieno[2,3-d]pyrimidine-6-carboxylic acid
2-[5-(1-cyclopropanecarbonylpiperidin-2-yl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(3-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-methylbutyl)-8-(oxolane-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(8-methylquinolin-5-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyridin-2-yl)piperazine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-methyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
1-(cyclopentylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-methoxy-1-[1'-(morpholine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(4aS,8aR)-6-(2,3-dihydro-1H-inden-2-yl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-{1-[(3,4-difluorophenyl)methyl]-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
5-[1-(cyclopropylmethyl)pyrrolidin-2-yl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]thiophene-2-carboxamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-hydroxyethyl)-3-{5-[(4-methyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
[(1,5-dimethyl-1H-indol-2-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(3S,4R)-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-({3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
4-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyridine
N-cyclopropyl-3-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]propanamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-(1H-pyrazol-1-yl)butanamide
N-{1-[1-(2-methanesulfonamidopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
5-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
N-methyl-4-[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
4-[(4-methanesulfonylphenyl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
[2-({4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-1-yl}methyl)phenyl]methanol
8-(3,6-dimethylpyrazin-2-yl)-1-oxa-8-azaspiro[4.5]decane
N-[3-(1H-indazol-1-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
N4,N4,N6-trimethyl-N6-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-4,6-diamine
(1S,5R)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
1-(furan-3-ylmethyl)-2-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
5-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-methoxy-4-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}pyridine-3-carbonitrile