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4-methyl-6-[3-(methylsulfanyl)phenyl]pyrimidin-2-amine
N-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]pyridin-3-amine
4-{[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-2-methylphenol
[1-(1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
8-{3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}-2,8-diazaspiro[4.5]decan-3-one
3-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
5-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-3-carboxamide
{[3-({1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(thiophen-3-ylmethyl)amine
1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperazin-2-one
(4aR,7aS)-1-(2-methoxyethyl)-4-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-5-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
5-{[2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamido]methyl}-N-methylfuran-2-carboxamide
1-tert-butyl-3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1H-pyrrole
2-[4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-ethylpiperidine-3-carboxylic acid
N-[1-(pyridine-4-carbonyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N4-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}pyrimidine-4,6-diamine
3-(4-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
1-[3-(1,2-oxazolidin-2-yl)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
(3R,4R)-1-[(3,5-difluorophenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
methyl 6-[(2-hydroxyphenyl)methyl]-2-[(4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-chlorophenyl)-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}cyclobutane-1-carboxamide
3-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
1-(2-methoxyethyl)-4-[({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)methyl]pyrrolidin-2-one
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
4-(4-chlorophenyl)-N-{[2-(3-acetamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}butanamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[2-(6-fluoro-2-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
2-(5-acetylthiophen-3-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
9-[(2S)-2-amino-2-cyclopropylacetyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methoxyethan-1-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
1-{1-[6-({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
ethyl 4-{[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]amino}piperidine-1-carboxylate
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
6-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N-ethylpyridine-3-carboxamide
2-fluoro-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
(2S,4S)-4-amino-1-(2-methoxybenzenesulfonyl)-N-methylpyrrolidine-2-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-ethyl-N-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
2-benzyl-4-[6-(trifluoromethyl)pyridin-3-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,5R)-3-(3-ethyl-1,2-oxazole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-2-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
9-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
1-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(2,3-dimethylphenyl)piperazine
1-({[(4-methyl-1,3-benzoxazol-2-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide