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N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-methyl-4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
2-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-2-(4-phenylpiperidin-1-yl)acetamide
1-[3-(1H-pyrazol-4-yl)benzoyl]-4-(thiophene-2-carbonyl)piperazine
(2S,4S)-1-benzyl-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-methylpyrrolidine-2-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]propan-1-one
1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
(3S,5R)-N3-(4-methylphenyl)-N5-(pyridin-3-ylmethyl)piperidine-3,5-dicarboxamide
4-{7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}-5-ethyl-6-methylpyrimidin-2-amine
(1R,5R)-6-(pent-2-yn-1-yl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}pyridin-1-ium-1-olate
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(quinoxalin-2-ylmethyl)acetamide
2-benzyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3-benzoxazole-5-carboxamide
2-(3-fluoro-4-methoxyphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
(2S)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-hydroxy-3-phenylpropan-1-one
1-{4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N'1-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N'1-methylcyclopropane-1,1-dicarboxamide
3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazine
2-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
methyl 2-(8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetate
[(2S,4R)-4-(dimethylamino)-1-(2-ethoxypyridine-3-carbonyl)pyrrolidin-2-yl]methanol
(4-{[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
2-methyl-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
methyl 8-[(3-methylphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,3-benzodiazol-2-yl]methanol
N,1-dimethyl-N-(quinoxalin-2-ylmethyl)azepane-2-carboxamide
3-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpropanamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-one
N-(3-hydroxypropyl)-1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-ol
ethyl 2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]amino}-1H-imidazole-5-carboxylate
4-methyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
1-(cyclohexylmethyl)-4-(2-methoxyethyl)-1,4-diazepan-5-one
2-(cyclopropylmethyl)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylazepan-3-amine
3-(3,4-dimethoxybenzoyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidine
1-{[(1H-1,3-benzodiazol-2-yl)carbamoyl]methyl}piperidine-3-carboxamide
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-methylpiperazin-2-one
4-(2-{1-[(4-methoxypyridin-2-yl)methyl]piperidin-2-yl}ethyl)phenol
2-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(propan-2-yl)pyrimidine
N-benzyl-5-fluoro-3-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-indole-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-(3-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propan-2-ol
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2-methyl-4-(2-methylphenyl)piperazine
N-methyl-N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}thian-4-amine
(3aS,6aR)-5-(pyrazin-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-1-(3-methylphenyl)urea
2-methoxy-1-[4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one