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4-[(benzyloxy)methyl]-1-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-(4-ethyl-1,4-diazepane-1-carbonyl)-8-methyl-2-(1H-pyrazol-4-yl)quinoline
ethyl({4-[2-(propan-2-yl)oxane-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)(pyridin-4-ylmethyl)amine
(1R,5S,6S)-N-methyl-3-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-N-(propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-[3-(benzyloxy)phenyl]-2-(carbamoylmethyl)piperidine-1-carboxamide
2-(4-fluorophenyl)-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2-methylpyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
8-[2-(3-fluorophenyl)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2R)-2-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-methylpentanamide
N-[2-(pyrazin-2-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-amino-6-(4-hydroxy-3-methoxyphenyl)-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
5-[3-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-oxopropyl]imidazolidine-2,4-dione
(3S,4R)-4-(4-fluorophenyl)-1-(2-hydroxyethyl)pyrrolidine-3-carboxylic acid
N,N-diethyl-1-({4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
3-[(3R,4S)-1-(2,6-difluoro-3-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-2-ol
(3aS,6aS)-2-acetyl-5-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-fluoro-1-(5-{1-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}thiophene-2-carbonyl)piperidine
1-{2-[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]ethyl}imidazolidin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(2,3,4-trifluorophenyl)ethan-1-one
5-methoxy-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-1H-indole-2-carboxamide
[(2-ethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
4-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
N-cyclopropyl-4-methoxy-2-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
ethyl 1-[1-(2-cyclopentyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperidine-2-carboxylate
N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(methylsulfanyl)ethyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
1-(2-{[(4-cyclopentylpyrimidin-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
9-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-2-amine
7-oxo-N-[(1-phenylcyclopentyl)methyl]-2-(pyridine-4-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,4-diazepane-6-carboxylic acid
2-acetyl-8-(quinolin-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyridin-2-ylmethyl)piperazine
2-(furan-2-yl)-5-{1-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
9-[2-(1H-imidazol-1-yl)propanoyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)sulfanyl]-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
4-benzyl-3-[1-(6-methylpyridine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2,5,6-trimethylpyrimidin-4-amine
N-({5-[(2,2-dimethyloxan-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N,N-dimethyl-2-{[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(3-hydroxy-3-phenylpyrrolidin-1-yl)-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
N-methyl-N-(propan-2-yl)-2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-acetyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
3-[2-(4-hydroxypiperidin-1-yl)ethyl]-8-methyl-3,4-dihydroquinazolin-4-one