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4-{[5-({[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}sulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine
1-amino-N-[(3R,4S)-4-(propan-2-yl)-1-(pyrimidin-2-yl)pyrrolidin-3-yl]cyclopropane-1-carboxamide
2-(1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-imidazol-2-yl)-1-methyl-1H-imidazole
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
5-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-acetamidoacetamide
1-phenyl-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperazin-2-one
5-methyl-1-[4-(pyridin-3-yl)pyrimidin-2-yl]-N-(quinolin-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-(1-ethyl-1H-1,2,3,4-tetrazol-5-yl)-1-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
N-[1-(4-chlorophenyl)cyclobutyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amine
3-[(5-ethylpyrimidin-2-yl)amino]-3-(4-methylphenyl)propan-1-ol
1-{3,9-diazaspiro[5.5]undecan-3-yl}but-3-en-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
2-cyclobutanecarbonyl-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(trimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methanol
2-{4-[2-(dimethylamino)phenyl]phenyl}-N-methylacetamide
3-cyclopropyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
5-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-4,6-dimethyl-2H-pyran-2-one
1-methyl-N-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-N-(pyridin-3-ylmethyl)piperidin-4-amine
6-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]pyridine-2-carboxylic acid
4-[(2-methylpyridin-3-yl)oxy]-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
ethyl 4-(2-phenylethyl)-1-(pyridine-4-carbonyl)piperidine-4-carboxylate
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
3-{5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
3-benzyl-4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-1-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-2-phenyl-N-[1-(1-propylpiperidin-4-yl)-1H-pyrazol-5-yl]acetamide
3-(cyclopropylmethyl)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidine-3-carboxylic acid
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-N-(4-methylphenyl)-2-oxoacetamide
N-[2-(oxolan-2-ylmethoxy)phenyl]-3-(pyridin-2-yl)azetidine-1-carboxamide
1-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
{1-[3-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)propyl]piperidin-3-yl}methanol
3-(piperidin-3-yl)-N-[3-(pyridin-3-yl)propyl]benzamide
1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]urea
3-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1H-indazole
N-cyclopentyl-2-{[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}propanamide
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
3-amino-1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}propan-1-one
[1-(diethylamino)propan-2-yl][(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
2-cyclopentyl-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}acetamide
2-methoxy-1-[4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3,3-dimethylcyclohexan-1-amine
N-(1-{[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
3-(1,3-benzothiazol-2-yl)-N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]propanamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,2,3-thiadiazole-4-carboxamide
3-(2-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}phenyl)pyrrolidine
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(2-aminoethyl)-1H-1,2,3-triazole-4-carboxamide
2-[9-(1H-indole-6-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide