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N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
9-(2-amino-2-methylpropanoyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-methoxy-1-methyl-2-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1H-indole
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-3-carboxamide
N4-(1,2-oxazol-3-ylmethyl)-7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(1-methoxypropan-2-yl)benzamide
1-(4-fluorophenyl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]cyclopropane-1-carboxamide
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
4-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,2-dimethylpiperazine
1-(6-ethyl-2-methylpyrimidin-4-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
methyl 2-[(1-methoxypropan-2-yl)sulfamoyl]-6-[3-(4-methylphenyl)propanoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{[2-(benzyloxy)phenyl]methyl}-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
1-(2-fluoro-4-methylbenzoyl)-4-(hydroxymethyl)azepan-4-ol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1H-imidazole-2-carboxamide
3-(2-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
(1S,5R)-3-(1H-indazole-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]furan-3-carboxamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1H-indazole-3-carboxamide
1-ethyl-6-[(4-methyl-3-phenylpiperazin-1-yl)methyl]-1H-indole
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-methoxy-5-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)pyrimidine
ethyl 1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-amido)piperidine-3-carboxylate
4-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-phenyl-1,3-oxazole
8-fluoro-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]quinoline-2-carboxamide
N-[2-(dimethylamino)ethyl]-5-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-2-methyl-1-benzofuran-5-carboxamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(dicyclopropylmethyl)methylamine
1-{3-[(3-chlorophenyl)methyl]-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(pyridin-4-ylmethyl)amine
(2S,4S)-4-[(dimethylcarbamoyl)amino]-N,1-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrrolidine-2-carboxamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-N-[1-(pyrazin-2-yl)propan-2-yl]piperidin-4-amine
7-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-(cyclobutylmethyl)-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-oxazepane
9-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-(cyclopropylsulfamoyl)-5-[4-(dimethylamino)phenyl]benzoic acid
2,3-dimethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-[(3-methoxyphenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
1-[4-(thiomorpholin-4-yl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
N-[3-(1H-indol-2-yl)phenyl]-1-(3-methylbutanoyl)piperidine-3-carboxamide
2-[5-(1,3-dimethyl-1H-pyrazol-4-yl)-1-(2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
(2S)-2-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-2-phenylacetamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
3-methyl-5-[1-({2-[(4-methylphenyl)methoxy]phenyl}methyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
5-(2,6-dimethylphenoxymethyl)-N-[2-(methylsulfanyl)ethyl]-1,2-oxazole-3-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide