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N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-6-[(4-phenylpiperidin-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
5-[(isoquinolin-5-yloxy)methyl]-N-(oxolan-3-ylmethyl)-1,2-oxazole-3-carboxamide
5-(3-fluorophenoxymethyl)-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-{4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[2-(4-chlorophenyl)ethyl]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
2-({[(3R,4R)-1-[(2,6-difluoro-3-methylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
3-(1-ethyl-1H-imidazol-2-yl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
6-methyl-2-(oxan-4-yl)-5-[5-(1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-[3-(1H-indol-3-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-2-(piperidin-1-yl)acetamide
2-{[2-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one
N-[(3R,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-2-carboxamide
7-hydroxy-4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-[4-(3-methoxyphenyl)phenyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-{2-[(1R,5S)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-(2-methyl-4-{[2-(pyridin-3-yloxy)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
methyl 4-(5-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-[2-(4-cyclohexyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-methyl-1,2-dihydrophthalazin-1-one
3-{2-cyano-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-N-(2-methylphenyl)-3-oxopropanamide
2-{4-[(4,4-difluoropiperidin-1-yl)methyl]-2-ethoxyphenoxy}propanoic acid
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-sulfamoylbutanamide
3-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-2-methylphenol
1-[2-(3-fluorophenyl)ethyl]-5-[4-(2-hydroxyethyl)piperidine-1-carbonyl]piperidin-2-one
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(5-ethylpyridin-2-yl)methyl]amine
(1S,5R)-3-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3,7-dimethyl-8-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
2-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-{[3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3,6-dimethyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-(2-ethylphenyl)-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
ethyl 5-{[cyclopropyl({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
2-[4-(methylsulfanyl)phenyl]-2-(pyrrolidin-1-yl)acetic acid
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}-1-phenylethan-1-ol
N-(3-hydroxy-3-methylbutyl)-N-methyl-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
6-methyl-4-(pyrrolidin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
3-phenyl-1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}pyrrolidin-3-ol
1-{4-[3-({[(4-methoxy-2,5-dimethylphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
N-[(2-ethoxyphenyl)methyl]-1-methylazepane-2-carboxamide
4-({[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
2-[(1S,5R)-3-(1H-indole-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(2-methoxyethyl)piperidine
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(4-methylphenyl)phenyl]piperidine-1-carboxamide