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5-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-1H-imidazole-4-carboxylic acid
2-(1-ethylpiperidin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
2-(3-fluoropyridin-4-yl)-8-methoxyquinoline
8-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[(2R)-2-aminopropanoyl]-N-[(4-chlorophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(1R)-1-(3-methoxyphenyl)ethyl]propanamide
3-({1-[(4-chlorophenyl)methyl]piperidin-3-yl}amino)-2,2-dimethylpropan-1-ol
3-phenyl-1-{1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propan-1-one
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(methylsulfanyl)ethan-1-one
4-[(2-chlorophenyl)methyl]-N-(2-ethylphenyl)-4-(hydroxymethyl)piperidine-1-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(1H-indazol-1-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide
5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazole
N-(2H-1,3-benzodioxol-5-yl)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
N-cyclooctyl-2-{[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]amino}acetamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-yl)pyridin-2-amine
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-3-(2-methylphenyl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]-2-(thiophen-3-yl)acetamide
2-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}pyridine
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(2,2,3,3-tetrafluoropropoxy)acetamide
2-[(2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
4-[(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
N,5-dimethyl-N-(1-methylpyrrolidin-3-yl)-2-phenylfuran-3-carboxamide
(4aR,7aS)-1-propanoyl-4-[(trimethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(propan-2-yl)-4-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]piperidine
N-ethyl-5-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]pyrimidin-2-amine
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]acetamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,2-dione
N-[(3S,4R)-1-(2-acetylbenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
9-[(3S)-3-hydroxy-3-phenylpropyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)cyclopropanecarboxamide
13-(2-chloro-4-fluorophenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-(oxan-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-methyl-2-(5-methyl-1H-pyrazol-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-ethyl-N,4-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,3-oxazole-5-carboxamide
N-(2-carbamoylethyl)-3-(3-chlorophenyl)-3-phenylpropanamide
3-chloro-5-({3-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
(3aS,6aR)-5-(piperidine-1-sulfonyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-{2-oxo-2-[3-(3-phenylpropanoyl)piperidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
3-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4H-chromen-4-one
4-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
2-(4-fluoro-3-methoxyphenyl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
2-{5-[(diethyl-1H-1,2,4-triazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
methyl 2-{7-chloro-3-[(2-methylpiperidin-1-yl)methyl]-2-oxo-1,2-dihydroquinolin-1-yl}acetate
4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2,3-dihydro-1H-imidazol-2-one
(3R,4R)-4-cyclopropyl-1-[(4-fluoro-3-methoxyphenyl)methyl]-3-methylpiperidin-4-ol
ethyl 3-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}propanoate