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3-methyl-1-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)butan-1-ol
N-[3-(furan-2-yl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
ethyl 1-[(4-methylthiophen-2-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(phenoxymethyl)pyrimidin-4-ol
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
4-({3-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenyl]phenyl}methyl)morpholine
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-2-oxo-2-(2-phenylindolizin-3-yl)acetamide
methyl 3-cyclobutaneamido-5-(cycloheptylamino)-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[(3-hydroxyphenyl)methyl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentyl-N-(2-methoxyethyl)-5-oxo-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxamide
1-{2-[(5-fluoropyrimidin-2-yl)oxy]hex-5-en-1-yl}-4-methyl-1,4-diazepane
2-methyl-4-(4-methylphenyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(6-methoxynaphthalen-2-yl)morpholine
1-cyclopentyl-4-{[2-(difluoromethoxy)phenyl]methyl}-1,4-diazepane
3-tert-butyl-1-methyl-4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-ethylpyrimidine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-1-benzofuran-5-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-[(3R,4S)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
6-methyl-5-{[4-(piperidine-1-carbonyl)piperidin-1-yl]methyl}quinoline
(3aS,6aR)-3-cyclopentyl-5-(4,4,4-trifluorobutyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
2-methoxy-5-methyl-N-{[1-(oxan-4-yl)piperidin-4-yl]methyl}benzamide
6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(3-methoxyphenyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclopentanecarboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(6-methoxypyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine-4-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-4-carboxylic acid
1-(3-methoxyphenyl)-5-methyl-4-[2-(phenylsulfanyl)acetyl]piperazin-2-one
4-(3-hydroxy-4-methoxyphenyl)-7-(2-oxopyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
6,7-dimethoxy-2-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-9-[6-(methoxymethyl)pyridine-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-(5-chloro-7-methoxy-1-benzofuran-2-amido)-N-ethyl-1-methylpyrrolidine-2-carboxamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-{[5-(1H-indol-3-ylmethyl)-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
4-{[2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-(2-hydroxypropyl)-9-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(3,3-diphenylpiperidine-1-carbonyl)-4-methyl-1,3-thiazol-2-amine
1-(3-ethyl-1H-indole-2-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
N-cyclopentyl-2-(dimethylamino)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)acetamide
N-[(5-fluoro-2-methylphenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-(4-hydroxy-3-methylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1S,3R)-3-amino-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)cyclopentane-1-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-4-(2-oxopyrrolidin-1-yl)benzamide
1-{1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperidin-4-yl}propan-1-ol
8-(2-hydroxyacetyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one