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2-(adamantan-1-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(methylsulfanyl)ethan-1-one
2-cyclopentyl-N-[3-(4-{[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
2-[benzyl(methyl)amino]-N-[2-(morpholin-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
7-[3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
6-(4-fluorophenyl)-N-methyl-N-[2-(piperidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
1-(2-methoxyacetyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-3-carboxamide
1-{4-[(1-hydroxyhexan-2-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-(1-propylcyclopropyl)-1-(pyridine-2-carbonyl)piperidin-4-amine
2-(5-{1-[6-(propan-2-yl)-1H-indole-2-carbonyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
4-cyclobutyl-2-(3-phenylpropyl)morpholine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]pyrazine-2-carboxamide
1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4-methylazepan-4-ol
4-[1-(methoxymethyl)cyclopropanecarbonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
3-benzyl-4-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-{2-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-1H-indole-3-carbonitrile
(2S,4R)-4-amino-N-ethyl-1-{3-[(4-fluorophenyl)formamido]propanoyl}pyrrolidine-2-carboxamide
6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
4-(5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
N,4-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
3-({1-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]propan-2-yl}oxy)pyridine
[1-(3-methoxybenzoyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(pyridin-3-yl)propyl]-1,2-oxazole-3-carboxamide
1-(3-{[5-methyl-6-(4-phenylazepane-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
2-{3-[(3-methoxyphenyl)methoxy]phenyl}-N-methylpyrimidin-4-amine
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
4-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,3-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-methanesulfonyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyrrolidine-2-carboxamide
N-benzyl-2-{3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
2-{3-cyclopentyl-5-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
(4aS,7aR)-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carbonitrile
2-(dimethylamino)-2-(4-methylphenyl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
(oxolan-2-ylmethyl)({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})(pyridin-2-ylmethyl)amine
methyl (2S)-2-cyclopropyl-2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}acetate
3-(morpholine-4-sulfonyl)-5-(pyridin-4-yl)benzoic acid
4-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-4-carbonyl}morpholine
1-[(2-fluorophenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-[4-(3-methylpiperidine-1-carbonyl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
1-(4-chlorophenyl)-N-({1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-methyl-8-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(2-methoxy-6-methylphenyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine-1-carboxamide