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N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]butanamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1,2,3,6-tetrahydropyridine
4-{[2-(dimethylamino)ethyl]amino}-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3,4-dihydropyrimidin-4-one
N,2,2,6,6-pentamethyl-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-4-amine
1-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidin-4-yl}pyrrolidin-2-one
N-propyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-methyl-1-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-(2-hydroxyethyl)-3-[(5-methylthiophen-2-yl)methyl]urea
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[3-(3-oxopiperazin-1-yl)propyl]acetamide
3-({1-[(3-methylthiophen-2-yl)sulfonyl]pyrrolidin-3-yl}methyl)benzamide
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-{4-oxo-3H,4H-pyrido[4,3-d]pyrimidin-3-yl}azepan-2-one
N-[(3S)-2-oxoazepan-3-yl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(4-methyl-1H-imidazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-benzyl-5-(5-cyclopropyl-1,3-oxazol-4-yl)-3-methyl-1H-1,2,4-triazole
N-cyclobutyl-7-[(2-methoxypyrimidin-5-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N5-cyclooctyl-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-N3-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethoxyphenyl)urea
1-amino-N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)cyclopropane-1-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
3-{1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
1-[1-(3-cyanobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
2-(3-chloro-4-fluorophenyl)-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
8-(1-hydroxypropan-2-yl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-fluorophenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-5-carboxamide
1-ethyl-N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1H-indole-5-carboxamide
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(naphthalene-1-carbonyl)piperidine
4-(cyclohexylmethyl)-3-{2-oxo-2-[4-(piperidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
6-chloro-N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
1-methoxy-3-{[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]amino}propan-2-ol
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[3-(pyridin-2-yl)propyl]propanamide
N-methyl-3-[(oxolan-3-ylmethyl)sulfamoyl]-N-(piperidin-4-yl)benzamide
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyridin-4-yl)-1,4-diazepane
1-({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrazol-1-yl)acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-ethyl-N,2-dimethyl-1,3-thiazole-5-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-ol
3-{[1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-3-yl]methyl}benzamide
[(3R,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[4-(2-methoxyquinolin-3-yl)-3,5-dimethyl-1H-pyrazol-1-yl]propan-2-one
(1s,4s)-4-{4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
2-(2-methoxyethyl)-5-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)pyrimidine
1-[2-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-({5-[(6-fluoroquinolin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea