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N-[(3S,5S)-1-cyclopentyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3,5-difluoropyridine-2-carboxamide
1-(2-{[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
2-(5-acetylthiophen-3-yl)-N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]acetamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-oxo-2-phenylacetamide
4-(1H-imidazol-1-yl)-1-(1-phenylcyclopropanecarbonyl)piperidine-4-carboxylic acid
2-(cyclohex-1-en-1-yl)-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]acetamide
4-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1,4-oxazepan-6-ol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
1-ethyl-N-[(3-fluorophenyl)methyl]-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(methylsulfanyl)propan-1-one
2-hydroxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
2-(2-ethylphenyl)pyridine-3-carbonitrile
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrrole-2-carboxamide
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methoxyphenyl)methyl]piperidine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
5-(1H-imidazol-2-yl)-1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazole
(3S)-N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-benzylpyrrolidin-3-amine
(2S)-1-[(4-{[2-(hydroxymethyl)phenyl]carbamoyl}phenyl)methyl]-N,N-dimethylpyrrolidine-2-carboxamide
2-fluoro-N-{1-[({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
4-(4-chlorophenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]butanamide
3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)benzonitrile
8-(1H-1,2,3-benzotriazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-(1-hydroxyhexan-2-yl)-2-(methylamino)pyrimidine-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}oxane-4-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-[(3-methylphenyl)methyl]piperazine
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
2-({[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-dimethoxyphenyl)acetamide
2-{5-[1-(2-hydroxyethyl)-4-phenyl-1H-imidazol-5-yl]furan-2-yl}benzonitrile
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
N-[3-(2-methylquinolin-4-yl)phenyl]acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{2-[(2-fluoro-5-methoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
4-chloro-1-methyl-3-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrazole
6-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
2-ethyl-5-{2-[2-(3-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
N-benzyl-3-(1,2-oxazinan-2-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
6-{[(4-methyl-1,4-oxazepan-6-yl)methyl]amino}pyridine-2-carbonitrile
(3S,4R)-4-(4-fluorophenyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-cyclohexyl-3-{[ethyl(pyridin-4-ylmethyl)carbamoyl]methyl}morpholine-4-carboxamide
8-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-5-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-[2-(azepan-1-yl)-2-oxoethyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide