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8-fluoro-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}quinoline-2-carboxamide
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2,2,2-trifluoroethyl)propanamide
5-[3-(piperidine-1-carbonyl)phenyl]furan-2-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
7-(3-chlorophenyl)-9-methoxy-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 2-(4-{[(2-fluoro-5-methylphenyl)carbamoyl]methyl}morpholin-3-yl)acetate
4-{4-ethyl-6-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidin-2-yl}morpholine
3-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
1-[(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
1-[(3-methoxyphenyl)methyl]-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidin-2-one
2-{5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
4-[4-(2,2-diphenylethyl)piperazin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
(2S,4R)-4-cyclopentaneamido-1-[(2,4-dimethylphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
(4aS,7aR)-1-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2S,4S)-1-(cyclohexylmethyl)-4-acetamidopyrrolidine-2-carboxylate
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
methyl 3-cyclohexaneamido-5-({[2-(methylsulfanyl)-1,3-thiazol-4-yl]formamido}methyl)benzoate
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine-4-carboxamide
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,3S,5S)-8-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
(1S,2R)-1-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}-2,3-dihydro-1H-inden-2-ol
9-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}ethan-1-one
[(3R,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]butanamide
2-(3-methyl-4-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
1-{1-[(2-ethoxynaphthalen-1-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
(2R,3R,6R)-5-(6-ethylpyrimidin-4-yl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[1-(cyclohexylmethyl)-4-(1H-indol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
3-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-1-(furan-2-ylmethyl)urea
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-hydroxyphenyl)-N-(2-methoxyethyl)acetamide
2-amino-6-cyclobutyl-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
4-{1-butyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl}benzamide
4-phenyl-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5-(thiophen-3-yl)-1H-imidazole
2-(3-fluorophenyl)-N-{[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
methyl (2S,4R)-1-[2-(cycloheptylcarbamoyl)ethyl]-4-hydroxypyrrolidine-2-carboxylate
1-cyclopropanecarbonyl-4-{4-[4-(3-methoxypropyl)piperidine-1-carbonyl]phenoxy}piperidine
(1S,5R)-6-methyl-7-oxo-N-[2-(trifluoromethyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)pyrrolidin-2-one
3-[(3-methoxypyrrolidin-1-yl)sulfonyl]-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
N-[2-(furan-2-ylmethoxy)phenyl]-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-4-carboxylate
1-({5-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
5-(4-acetylphenoxymethyl)-N-(2-methylpropyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
(2R,3R)-3-amino-1'-(pyridin-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-chloro-2-[2-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-1H-pyrrol-1-yl]pyridine
methyl 7-oxo-9-(propan-2-yloxy)-3-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(furan-2-yl)ethyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide