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(3aR,5R,6S,7aS)-2-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-octahydro-1H-isoindole-5,6-diol
N-[3-(1,2,3,4-tetrahydroisoquinolin-7-yl)phenyl]acetamide
(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
1-(isoquinoline-3-carbonyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-[(3R,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
4-(3-{[4-(piperidin-1-yl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
N-(naphthalen-1-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
1-[2-(3-methoxyphenyl)piperidin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-phenyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
1-(2-methoxyethyl)-4-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
(4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}morpholin-3-yl)methanol
2-{4-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-[(3,4-difluorophenyl)methyl]-3-[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]propanamide
(2S,4S)-N-ethyl-4-[2-(2-fluorophenyl)acetamido]-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxamide
5-methoxy-N-methyl-N-[1-(pyridin-4-yl)ethyl]furan-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}pyridine-3-carboxamide
2-[2-(3,4-difluorophenyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[6-(hydroxymethyl)pyridine-2-carbonyl]pyrrolidin-3-yl]methanol
N-(3-benzylphenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]piperidine-3-carboxamide
1-(2-{3-cyclopropyl-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3,5-dimethylphenyl)-1H-pyrazole
N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(3-hydroxyphenyl)methyl]acetamide
N-propyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl][2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]methylamine
N-[3-(3-fluorophenyl)phenyl]-1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide
ethyl 1-(1-{[7-fluoro-2-oxo-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperidin-4-yl)piperidine-3-carboxylate
5-ethyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]thiophene-2-carboxamide
8-(4-acetylbenzoyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-[4-(4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
7-(3-chlorophenyl)-4-(3-fluoropyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-6-{[2-(difluoromethoxy)phenyl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
8-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}-2,8-diazaspiro[4.5]decan-3-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(1,2-oxazinan-2-yl)propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridine
3-(2-methylpropyl)-6-[(3,4,5-trimethoxyphenyl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1-hydroxypropan-2-yl)acetamide
2,2-diethyl-4-[4-(piperidin-3-ylmethyl)benzoyl]morpholine
2-[4-chloro-2-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)phenoxy]acetic acid
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
(4S)-3,3,4-trimethyl-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-ol
N-(1-{[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
1-[(1S,5R)-6-(2,3,4-trifluorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[(3-methylthiophen-2-yl)methyl]-1,1-dioxo-N-(pyridin-2-ylmethyl)-1λ6-thiolane-3-carboxamide