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2-(2-fluoro-6-methoxyphenyl)-N-methylpyridine-3-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
methyl 4-{3-[1-(furan-3-ylformamido)-2-methylpropyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}benzoate
N-(propan-2-yl)-5-(pyrimidin-5-yl)furan-2-carboxamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-5-propyl-1,2-oxazole-3-carboxamide
N-(1-{7-[(8-methoxyquinolin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-cyclopentyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-(1H-imidazol-2-yl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
1-(cyclopropylmethyl)-5-(2-methoxypyridine-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)propanamide
1-[3-(2-methylphenyl)phenyl]-N-(piperidin-4-ylmethyl)piperidin-4-amine
2-cyclobutyl-N-[(3R,4S)-4-propyl-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]acetamide
1-(5-{[4-(ethylamino)pyrimidin-2-yl]amino}-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
N-{[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
1-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-methoxy-1-{4-[4-(1,2-oxazinane-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-[4-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-(2-hydroxyethyl)-5,6-dimethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
9-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-diethyl-3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
N-(1-phenylcyclopropyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-ethyl-3-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
N'-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N,N-dimethylbutanediamide
5-ethyl-1'-[(8-fluoroquinolin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 4-benzyl-1-[(3,5-difluorophenyl)methyl]piperidine-4-carboxylate
3-(4-hydroxyphenyl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
8-[(5-chlorothiophen-2-yl)methyl]-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclopentyl-N-ethyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
3-{5-[1-(2-phenylethyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
5-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(2-methylpropyl)-1H-imidazole
{1-[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl]piperidin-4-yl}(pyridin-2-yl)methanol
(3R,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidin-3-amine
5,7-dimethyl-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
2-amino-N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-4-methylpyrimidine-5-carboxamide
N-[3-(4-{[3-(1H-imidazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
N,1,6-trimethyl-N-(3-phenylpropyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
1-(5-{[(furan-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
4-{4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-{2-[2-(furan-2-yl)-2-oxoacetamido]-5-methoxyphenyl}-2-methylpropanamide
4,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
N'-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-N-(5-methyl-1,2-oxazol-3-yl)ethanediamide
N4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine