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1-(6-ethoxy-4-methylquinazolin-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-2-carboxamide
5-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
(3R)-1-[(4-methoxypyridin-2-yl)methyl]-3,4,4-trimethylpyrrolidin-3-ol
1-{4-[1-(2-methoxyethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}butan-2-ol
1-{2-[3-(methanesulfonylmethyl)piperidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(propan-2-yloxy)-N4-(pyridin-2-ylmethyl)pyrimidine-2,4-diamine
N-[(2R)-1-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1-oxopropan-2-yl]acetamide
N-(2-aminoethyl)-3-({[3-(1H-pyrazol-1-yl)phenyl]methyl}sulfamoyl)benzamide
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
2-phenyl-1-{4-[2-(3-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
2-(2-chloro-4-fluorophenyl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]acetamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidine-1-carbonyl)pyrazine
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pentanamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-(2,6-dimethylpyridin-3-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)pyrimidin-2-amine
4-{[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]amino}-2-methylpentan-2-ol
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-cyclopropanecarbonylpiperidine
N-cyclopentyl-6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
[(3aS,6aS)-2-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-methyl-5-oxo-1-(pyridin-2-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxamide
3-({[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]amino}methyl)piperidin-3-ol
5-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-ethoxy-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylpyrimidin-2-amine
4-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-3-cyclobutyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(propan-2-yl)-2-(1-propylpiperidin-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-[3-(dimethylcarbamoyl)-4-methoxyphenyl]-4-(pyridin-3-yl)piperazine-1-carboxamide
7,7-dimethyl-2-[1-(2-phenylethyl)piperidin-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[benzyl(methyl)amino]-3-(4-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
ethyl 3-[(3-chlorophenyl)methyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-3-carboxylate
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[3-(1H-indol-1-yl)propyl]acetamide
2-{2-[(dimethylamino)methyl]phenyl}-N-ethylpyrimidin-4-amine
8-[(4-carboxyphenyl)methyl]-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
2,6-difluoro-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}benzamide
2-(2-methyl-1,3-thiazol-4-yl)-5-[4-(propan-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
1-(2-methyl-1-benzofuran-5-carbonyl)-4-phenylpiperidine-4-carbonitrile
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(1H-indol-3-yl)-N-methylpropanamide
2-[(4aS,7aR)-4-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N,1-dimethyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(methylamino)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2,5-dimethyl-3-[4-(oxolan-3-ylmethyl)piperazin-1-yl]pyrazine
4-{[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]amino}-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
3-(4-tert-butylbenzoyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(3-chlorophenyl)ethyl]piperidine-4-carboxamide
3-{4-phenyl-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-5-yl}quinoline