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[7-(1,3-benzothiazol-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
4,6-dimethyl-3-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(3S)-1-(1-methyl-5-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-1H-1,3-benzodiazol-2-yl)pyrrolidin-3-ol
5-ethyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-methylpyrimidin-4-amine
4-(4-methyl-1H-pyrazol-1-yl)-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidine-4-carboxylic acid
N-[2-(2-methyl-1-phenyl-1H-indol-3-yl)ethyl]-3-(2-methyl-5-oxopyrrolidin-2-yl)propanamide
methyl 4-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-4-oxobutanoate
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
6-methyl-2-[1-(3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[(2-phenoxypyridin-3-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
methyl 4-{4-[(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-5-methyl-1,3-oxazol-2-yl}benzoate
2-methoxy-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
2-(6-aminopyridin-3-yl)-2-{[(8-methoxyquinolin-5-yl)methyl](methyl)amino}acetic acid
2-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-6-fluoroquinolin-4-ol
4-{5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
6-(2-methoxypyridin-3-yl)-1H-1,3-benzodiazole
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3,6-dimethylpyrazin-2-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperazine-1-carboxamide
7-(2,6-dimethylhept-5-en-1-yl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-[(3-methoxyphenyl)methyl]-4-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]morpholine
(1S,5R)-6-(5-fluoropyridine-3-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(3S,4S)-1-(furan-2-ylmethyl)-4-[4-(pyridin-3-yloxy)piperidin-1-yl]pyrrolidin-3-ol
N-(pyridin-3-ylmethyl)-1-[1-(4,4,4-trifluorobutyl)piperidin-4-yl]piperidine-4-carboxamide
(2S)-3-phenyl-2-{[3-(1H-pyrazol-4-yl)phenyl]formamido}propanamide
11-{[(3-chlorophenyl)methyl]amino}-4-(3-methylbutyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(5-methylthiophen-2-yl)-N,N-bis(prop-2-en-1-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2,6-dihydroxy-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}benzamide
2-methyl-N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-1-phenyl-1H-1,3-benzodiazole-5-carboxamide
(3S,4S)-1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
1-(2-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
4-(5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)pentan-1-one
1-[4-({[(2,5-dimethoxyphenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
4-(1H-pyrazol-1-yl)-1-(quinoxaline-6-carbonyl)piperidine-4-carboxylic acid
5-ethyl-4-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]pyrimidin-2-amine
2-(2-oxopyrrolidin-1-yl)-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)acetamide
2-chloro-N-[2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-methoxy-6-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
4-(5-acetyl-4-methylpyrimidin-2-yl)-N,N-dimethylpiperazine-1-sulfonamide
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-methylurea
3-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-[(1R,5S)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
ethyl 4-[({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)methyl]-1H-pyrazole-3-carboxylate