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N-(adamantan-1-yl)-6-{[benzyl(butyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{3-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-ol
N-[2-(3-methoxyphenyl)-1-{1-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
1-(3-chlorophenyl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperazin-2-one
(3-{2-[1-(2,4-difluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-cyclopropyl-6-oxo-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-5-methylpyridine-3-carboxamide
2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
N-cyclohexyl-N-(pyridin-3-ylmethyl)morpholine-2-carboxamide
2-[2-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)-4-(thiophen-2-yl)phenoxy]acetic acid
3,5,7-trimethyl-2-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-indole
6-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-fluoro-5-{[(1-methanesulfonylpiperidin-4-yl)carbamoyl]amino}benzamide
N-methyl-N-{2-phenyl-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl}pyridine-2-carboxamide
1-ethyl-N-methyl-5-({[1-(piperidin-1-yl)cyclohexyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
(1R,7S)-N-(2-hydroxyethyl)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 2-[(2R,3R)-2-hydroxy-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]acetate
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]urea
N2,N2,N4,5,6-pentamethyl-N4-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]acetamide
4-{3-[3-(3-methoxybenzoyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(3-methylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-hydroxy-1-{[5-(methylcarbamoyl)thiophen-3-yl]sulfonyl}piperidine-4-carboxylic acid
1-[(2-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
5-ethyl-2,3-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(3aR,6aR)-3a-(4-propyl-1,4-diazepane-1-carbonyl)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methoxyethan-1-one
2-[5-(methoxymethyl)-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
2-{1-[(4-fluorophenyl)methyl]-4-[(2-methyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
7-fluoro-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-[2-(3-phenylpropoxy)phenyl]-4H-1,2,4-triazole
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(morpholin-3-yl)acetamide
3-(2-methoxyethyl)-1-(3-methoxypyrazin-2-yl)piperidine-3-carboxylic acid
3-methyl-8-[2-(3-methylphenyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-propyl-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-[1-(pyrazin-2-yl)propan-2-yl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazole
4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}pyrimidine
1-{4-[(4-methyl-3-phenyl-1,2-oxazol-5-yl)amino]piperidin-1-yl}ethan-1-one
N-cyclohexyl-1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
(3R,4R)-4-(azepan-1-yl)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-ol
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(4,4,4-trifluorobutyl)piperidine
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(5-methylpyrazin-2-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-amino-4-(2-methyl-1H-imidazol-4-yl)-5H-chromeno[4,3-b]pyridine-3-carbonitrile
N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-{[(3R,4R)-4-(hydroxymethyl)-1-(9H-purin-6-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol