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[4-propoxy-3-(pyrimidin-5-yl)phenyl]methanol
(4aR,7aS)-1-cyclobutanecarbonyl-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
N,N-dimethyl-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine-1-sulfonamide
2,6-dimethyl-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyrimidine-4-carboxamide
5-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenylethane-1,2-dione
N-(2-hydroxy-3-methoxypropyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-[2-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-4-methanesulfonylpiperazine-1-carboxamide
1-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
2-methoxy-3-[1-methyl-5-(morpholin-4-yl)-1H-1,2,4-triazol-3-yl]quinoline
1-[3-(2-methylphenyl)piperidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(2,6-dimethylpyridine-4-carbonyl)-4-(thian-4-yl)piperazine
3-{[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}azepan-2-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
2-amino-2-methyl-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
9-(dimethyl-1,3-oxazole-5-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3-chlorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
3-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-N-(2,2,2-trifluoroethyl)benzamide
1-(cyclohexylmethyl)-N-methyl-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzonitrile
1-{2-[2-(1-methylpiperidin-4-yl)-1H-imidazol-1-yl]ethyl}-3-phenylpiperidine
1-(4-butyl-6-hydroxy-1,4-diazepan-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
(4aR,7aS)-N,N-dimethyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
9-methoxy-7-(5-methylthiophen-2-yl)-4-(1H-1,2,4-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-(1H-imidazol-1-ylmethyl)piperidine
[(2-fluorophenyl)methyl](2-methoxyethyl)(quinolin-2-ylmethyl)amine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethyl}pyrrolidin-2-one
5-oxo-N-[3-(pyridin-2-yl)propyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
[3-(1-methyl-1H-pyrazol-4-yl)-4-propoxyphenyl]methanol
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[2-(2-phenylethyl)morpholin-4-yl]ethan-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-(2-methylphenyl)-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}acetamide
N4-ethyl-N2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
(4aS,8aR)-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
N-(cyclopropylmethyl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
N-cyclopentyl-2-({[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}amino)butanamide
2-[benzyl({[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
2-[(3,5-difluorophenyl)methyl]-8-(3-fluoropyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
5-(2-fluorophenyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-4-sulfamoylbenzamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
(3S,4S)-1-(6-aminopyridine-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol