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7-methoxy-3-{[2-(trifluoromethyl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-N-[2-(methylsulfanyl)phenyl]propanamide
1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3-(thiophene-2-carbonyl)piperidine
3-chloro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
6-cyano-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyridine-3-carboxamide
1-[1-(2-aminoacetyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(3-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
4-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-2-yl}-2-methoxyphenol
4-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
3,6-dimethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
7-[(3,4-difluorophenyl)methyl]-2-methyl-2,7-diazaspiro[4.5]decan-6-one
8-{6-azaspiro[2.5]octane-1-carbonyl}-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-ethyl-3-(pyrrolidine-1-carbonyl)-N-(quinolin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclopropanecarboxamide
N-(1-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
N-{[3-(difluoromethoxy)phenyl]methyl}-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-acetyl-N-(2H-1,3-benzodioxol-5-ylmethyl)-2,4-dimethyl-N-(propan-2-yl)-1H-pyrrole-3-carboxamide
1-[(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
(4aR,7aS)-1-acetyl-4-[(3-chlorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-({1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]azepan-3-yl}amino)pyridine-2-carbonitrile
7-chloro-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-methyl-1H-indole-2-carboxamide
4-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-2-[2-(3-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
3-methyl-3-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)-1λ6-thiolane-1,1-dione
8-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
1-{2-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,3-benzotriazole
(2R,6S)-2,6-dimethyl-4-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}morpholine
(3R,5S)-5-[1-(4-fluorophenyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol
N-[3-(methylsulfanyl)propyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}piperidin-2-one
1-(7-methyl-3-{[(2-methylpropyl)amino]methyl}quinolin-2-yl)piperidin-4-ol
4-[(diethylamino)methyl]-5-ethyl-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}furan-2-carboxamide
2-ethoxy-6-{[methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
6-(4-acetyl-1,4-diazepan-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
7-(3-chlorophenyl)-4-(pyrrolidine-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclohexyl-4-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
4-cyclobutyl-6-methyl-2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyrimidine
6-methyl-2-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}methyl)-1H-1,3-benzodiazole
2-[(3-{[2-(pyridin-3-ylformamido)ethyl]carbamoyl}phenyl)amino]acetic acid
1-(2-propoxyethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(3R,4S)-3-amino-4-(2-hydroxyethyl)pyrrolidin-1-yl]-2-(2,4-dichlorophenoxy)ethan-1-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-4-methyl-2-(methylamino)-1,3-thiazole-5-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-(6-methylpyrimidin-4-yl)piperidine-4-carboxamide
4-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-8-fluoroquinoline-2-carboxamide
(1S,5R)-6-propyl-3-[3-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one