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1-[3-(3-chlorophenyl)phenyl]-3-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}urea
1-[1-(3-chlorobenzoyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
3-(2-methylphenyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
9-(2-ethoxyethyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(1H-imidazol-1-yl)butan-2-yl]-N'-[2-(propan-2-yl)phenyl]butanediamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2,5-dimethylpyrimidine
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
2-methyl-4-{4-[3-(pyridin-2-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
(2S)-2,6-diamino-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)hexanamide
N-[(3R,5S)-1-(cyclopentylmethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
4-(4-tert-butylphenyl)-3-(4-methyl-1H-imidazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-ethoxypyridin-3-yl)methyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
9-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
9-methyl-3-(5-propylpyrimidin-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
(3S,5R,9R)-5-hydroxy-11-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[2-(propylsulfanyl)phenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
ethyl 4-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazine-1-carboxylate
1-[(1S)-1-phenylpropyl]-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
3-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
5-amino-3-(3,4-dihydroxyphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)-1,3-benzoxazole
8-[3-(2-methylpropyl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl]quinoline
4-(1H-imidazol-2-yl)-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
5-(3-acetylphenoxymethyl)-N-methyl-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
3-benzyl-5-(3-methylfuran-2-yl)-1H-1,2,4-triazole
2-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-5-propylpyrimidin-4-amine
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-2-methanesulfonylacetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
N'-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]butanediamide
N-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1H-indazole-3-carboxamide
N-(1-carbamoylcyclopentyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N6-methyl-N6-[(trimethyl-1H-pyrazol-4-yl)methyl]-9H-purine-2,6-diamine
N2,N4-dimethyl-N2-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-2,4-diamine
6-ethyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrimidin-4-amine
5-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methoxy-3-[3-(pyridin-4-yl)azetidin-1-yl]pyrazine
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3,5-difluoro-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-{1-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
(2S)-2-amino-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-phenylacetamide
5-{2,6-dimethylimidazo[1,2-a]pyridin-3-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
methyl 3-({[1-(oxan-4-yl)piperidin-4-yl]carbamoyl}amino)benzoate
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
N-{[3-(dimethylamino)phenyl]methyl}-5-methoxy-1-methyl-1H-indole-2-carboxamide