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4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
1-(2-methoxy-5-{[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
4-[(furan-2-ylmethyl)amino]-N,5-dimethyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxamide
7-[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]-5-phenylpyrazolo[1,5-a]pyrimidine
N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-4-(thiophen-2-yl)butanamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}propanamide
N-cyclopentyl-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[3-methoxy-4-(oxan-2-ylmethoxy)phenyl]methyl}benzamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-3-(1H-pyrazol-1-ylmethyl)benzamide
(2S,4S)-4-(2,5-dimethylfuran-3-amido)-N-ethyl-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
2-(3-methoxyphenyl)-N-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]azetidine-1-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-methyl-N-(oxan-4-yl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}isoquinoline
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
N-{2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-oxoethyl}methanesulfonamide
ethyl 4-(2-phenylethyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-4-carboxylate
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
4-[(3-hydroxyphenyl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,5-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
1-[(2S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
3-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}-1-(4-methylpiperidin-1-yl)propan-1-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
N5-cyclooctyl-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N3-[3-(3-ethylphenoxy)propyl]-N3-methylpiperidine-1,3-dicarboxamide
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-methyl-N-(oxan-4-yl)-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
9-[2-(4-chloro-2-methylphenoxy)acetyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
4-(1-methyl-1H-pyrazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-benzyl-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrrolidin-2-one
ethyl 5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(2,3-dihydro-1H-indol-1-yl)-2-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}ethan-1-one
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
2-{3-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-[(3-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-({[3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
6-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-ethyl-6-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-4H-pyran-2-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-bromobenzamide
7-(dimethylamino)-4-[3-(morpholin-4-ylmethyl)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
(1S,5R)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-[5-(2-ethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
8-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-8-fluoroquinoline-2-carboxamide