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2-[2-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]ethan-1-ol
N-{[1-(3-chlorophenyl)pyrrolidin-3-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
(3S,4S)-1-(5-ethylpyrimidin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
5-(2,6-dimethoxyphenyl)-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1,2,4-triazin-3-amine
3-(azocan-1-yl)-N-(1-benzylpiperidin-4-yl)propanamide
5-[1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)pyrrolidin-2-yl]-3-methyl-1,2-oxazole
1-(2-oxo-2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}ethyl)pyrrolidin-2-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-methyl-1,3-benzoxazole-6-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carboxamide
1-[(2-methoxyphenyl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
1-[(2,3-difluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-methyl-4-(5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carbonyl)piperazin-2-one
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-3-ol
[1-({1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
4-(8-methoxyquinolin-5-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(2R)-2-amino-1-[4-(2,2-dimethoxyethyl)piperazin-1-yl]-2-phenylethan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-methylphenyl)-3-phenylpropanamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(3,4-difluorophenyl)methyl]piperidine
2-{[4-(3-acetylphenyl)-5-cyclopropyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-ethyl-3-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-{4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
5-{[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-benzyl-1-cycloheptyl-6-oxopiperidine-3-carboxamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-ol
ethyl 1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-{5-[2-(dimethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-4-phenylazepane-1-carboxamide
3-{4-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
4-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidine-4-carbonyl}morpholine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-yl]methanol
3-[(1-ethyl-1H-indol-5-yl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-cyclooctyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(ethylsulfanyl)-5-{[(2S)-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]methyl}pyrimidine
3-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]sulfonyl}-N-cyclobutylbenzamide
1-{2-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-4-methylpyrimidin-5-yl}ethan-1-one
4-(3-chlorophenyl)-5-(methoxymethyl)-3-methyl-1H-pyrazole
4-{4-[4-(2-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]pyridine
5-cyclopropanecarbonyl-1'-(2,3-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-3-(5-methylfuran-2-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
6-{3-oxo-3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
(2-methylpropyl)({[1-(propan-2-yl)piperidin-4-yl]methyl})(pyridin-2-ylmethyl)amine
3-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
1-[(2-methoxyphenyl)methyl]-5-(morpholine-4-carbonyl)piperidin-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(trifluoromethyl)benzamide