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1-(6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-yl)ethan-1-ol
(2S)-1-(benzylsulfamoyl)-N-ethylpyrrolidine-2-carboxamide
1-(4-fluoro-3-methoxyphenyl)-3-[3-(3-oxopiperazin-1-yl)propyl]urea
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)thiophene-3-carboxamide
1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-[5-(1-ethylpyrrolidin-3-yl)-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]pyridine
N-[(5-fluoro-1H-indol-2-yl)methyl]-6-(methoxymethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}(4,4,4-trifluorobutan-2-yl)amine
4'-(4-phenoxybutyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}-1,4-oxazepan-6-ol
3-{1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
N,N-diethyl-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}urea
4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
1-(4-ethylpiperazin-1-yl)-3-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}propan-1-one
N-[2-(3-phenylpiperidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
1-(3-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-[2-(4-methylmorpholin-2-yl)ethyl]-3-(2-methylphenyl)propanamide
(4aR,8aS)-6-(2-cyclopentylacetyl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
3-(2-methylphenyl)-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
N-(3-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-oxopropyl)acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-[(4-methanesulfonylmorpholin-2-yl)methyl]propanamide
5-(1-ethyl-1H-imidazol-2-yl)-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
8-(1,3-benzothiazol-2-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]acetamide
1-ethyl-3-(4-methoxy-3-methylphenyl)-N,N-dimethyl-1H-1,2,4-triazol-5-amine
4-[1-benzyl-5-(1-methylpiperidin-3-yl)-1H-1,2,4-triazol-3-yl]pyridine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(2-methyl-1H-imidazol-1-yl)propanamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-4-(1H-indol-3-yl)butan-1-one
1-[2-(2-fluorophenyl)ethyl]-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
N-[(3S,5S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-2-carboxamide
1-ethyl-8-{[3-(2-methylphenyl)phenyl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(2-methoxyphenyl)-3-methylpentyl]-2-methyl-1,3-thiazole-4-carboxamide
3-[2-({[(2S)-5-oxopyrrolidin-2-yl]methyl}(pyridin-2-ylmethyl)amino)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
{[1-benzyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]methyl}urea
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}pyrrolidin-2-one
2-(4-{[2-(cyclohex-3-en-1-yl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-ol
1-[3-(furan-2-yl)-5-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[(3-methylpyridin-4-yl)methyl]benzamide
2-(dimethylamino)-2-(2-methylphenyl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]acetamide
3-[(3R,4S)-4-(dimethylamino)-1-{2-[(2-methylphenyl)sulfanyl]acetyl}piperidin-3-yl]propanoic acid
2-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-1,3-thiazole
(1R,5S,8S)-8-hydroxy-N-(1-methyl-1H-indazol-5-yl)-3-azabicyclo[3.2.1]octane-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-(3-propylmorpholin-4-yl)ethan-1-one
(3R,4S)-3-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetamido]-4-cyclopropyl-N,N-dimethylpyrrolidine-1-carboxamide
6-(4-methyl-3-phenylpiperazin-1-yl)-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-hydroxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one