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4-[1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]thiomorpholine
4-[(4-ethyl-5-methylpyrimidin-2-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
1-butyl-3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-1-[(5-methylthiophen-2-yl)methyl]urea
8-methyl-2-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decane
3-hexyl-8-(2-hydroxy-3-methylbutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
1-(2-methylpropyl)-4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrrolidin-2-one
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}furan-2-carboxamide
methyl 4-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
8-(2-amino-6-methylpyrimidin-4-yl)-3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]quinoline-4-carboxylic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
2-methyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-1,3-benzodiazole
N-(1,3-benzothiazol-5-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
3-(1,2-oxazinan-2-yl)-N-[3-(propan-2-yloxy)propyl]propanamide
(2S,4S)-4-amino-N-methyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide
{3-[(3-methoxyphenyl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methanol
4-(3-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}phenyl)phenol
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]thiomorpholine
4-(4-{2-[(4-fluoropiperidin-1-yl)methyl]phenoxy}butyl)morpholine
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-(furan-2-ylmethyl)pyridine-2-carboxamide
1-(azepan-1-yl)-3-[4-({[(3,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-({4-hydroxy-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]azepan-4-yl}methyl)methanesulfonamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
5-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2,1,3-benzoxadiazole
2-(cyclopent-1-ene-1-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
ethyl 4-(cyclopropylmethyl)piperidine-4-carboxylate
N-[5-(pyrimidin-5-yl)quinolin-8-yl]acetamide
3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-N-ethylacetamide
N-{1-[1-(2-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
methyl 2-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
1-[(4aR,8aS)-1-[2-(2,3-difluorophenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
4-{2-[1-(1-aminocyclopropanecarbonyl)piperidin-2-yl]ethyl}phenol
3,3-dimethyl-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}cyclohexan-1-amine
2-(1-benzofuran-2-yl)-1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazole
4-(1-{2-[methyl(propan-2-yl)amino]acetyl}piperidin-3-yl)benzoic acid
1-methyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperazine
2-phenoxy-N-(4-{4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]piperidin-1-yl}phenyl)acetamide
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(3-methoxyphenyl)methyl]piperidin-4-ol
2-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}amine
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-methyl-3-(2-oxopyrrolidin-1-yl)-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]propanamide
N-cyclopropyl-4-{[2-(1,3-thiazol-4-yl)ethyl]sulfamoyl}benzamide