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5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-(2,5-dioxoimidazolidin-4-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)propanamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
1-(cyclohexylmethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
1-(2-methylphenyl)-3-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(3S,4S)-1-[2-methyl-2-(morpholin-4-yl)propanoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-[4-(propan-2-yloxy)phenyl]acetic acid
N-(1-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}cyclopentyl)aniline
N-[2-(4-methylpiperazin-1-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
6-(4-hydroxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(thiophen-2-yl)acetamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(quinolin-5-ylmethyl)piperidin-3-yl]propanamide
N-[2-(butan-2-yloxy)phenyl]-4-(2-methanesulfonylethyl)piperazine-1-carboxamide
1-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]pyrrolidin-2-one
N-({7-[2-(2-chloro-6-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
1-cyclopentyl-4-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-{4-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
dimethyl[(4-{1-[(1-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}phenyl)methyl]amine
2-methyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(3S,4R)-1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3-methoxypiperidin-4-amine
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl})methylamine
2-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzonitrile
2-methyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]furan-3-carboxamide
6-ethyl-2-methyl-N-(1-phenylpiperidin-4-yl)quinoline-4-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(piperidin-1-ylmethyl)piperidine
N-cycloheptyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl](methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
(4aS,8aR)-6-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
9-[2-(4-fluoro-2-methylphenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(6-methyl-2-propylpyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
3-(2-methoxybenzoyl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
2-(4,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
methyl({2-phenyl-1-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl})(pyridin-4-ylmethyl)amine
6-fluoro-2-({[(2S)-1-hydroxypropan-2-yl]amino}methyl)quinolin-4-ol
N-(butan-2-yl)-5-(3-cyanophenyl)furan-2-carboxamide
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
2-(2,6-dimethoxy-4-methylphenyl)-N-methylpyrimidin-4-amine
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-3-carboxamide
1-(furan-2-carbonyl)-4-(1,2-oxazole-3-carbonyl)piperazine
[(4-ethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-[1-(4-carbamoyl-1,3-thiazol-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
(4-{[1-(5-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-{2-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
4-(quinolin-4-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[4-(trifluoromethoxy)phenyl]methyl}cyclopropanamine
ethyl 4-[(3-methoxyphenyl)methyl]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine-4-carboxylate
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-5-phenylpentane-1,5-dione