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8-[5-(hydroxymethyl)furan-2-carbonyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-{[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}propanamide
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[(2,2-dimethyloxan-4-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
methyl(naphthalen-1-ylmethyl)[(3-{2-[4-(pyridine-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
2-(1-ethylpiperidin-4-yl)-1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}ethan-1-one
(1R,5S,8S)-8-methoxy-3-[3-(pyrrolidine-1-carbonyl)benzenesulfonyl]-3-azabicyclo[3.2.1]octane
8-methyl-N-[(4-methylpyridin-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(dimethylamino)ethan-1-one
N-methyl-2-[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-(propan-2-yl)acetamide
methyl 5-cyano-2-methyl-6-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyridine-3-carboxylate
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-7-oxo-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(morpholin-3-yl)acetamide
(3S,4R)-3-[(dimethylsulfamoyl)amino]-N-(2-fluorophenyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide
2-[1-(thiophen-2-ylmethyl)-4-[3-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]ethan-1-ol
N-[(3S,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
(3S,4S)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
6-(4-chloro-1H-indazol-1-yl)pyridin-2-amine
N-({3-[3-(pyridin-4-yl)propoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-(trifluoromethoxy)benzene-1-sulfonamide
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2,5,6-trimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrimidin-4-amine
4-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}piperazin-2-one
6-ethyl-2-methyl-4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}quinoline
8-[(dimethyl-1,3-thiazol-5-yl)sulfonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-(prop-2-en-1-yl)urea
N-{3-[(pyridin-3-yl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5R)-6-[2-(benzyloxy)ethyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
2-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]azetidin-3-yl}-1H-1,3-benzodiazole
1-{5-[4-(thiomorpholine-4-sulfonyl)phenyl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
2-{1-[(3,4-difluorophenyl)methyl]-4-(2,3-dihydro-1H-inden-2-yl)piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-(4,4,4-trifluorobutyl)pyrrolidin-3-yl]-1-ethyl-1H-pyrazole-5-carboxamide
4-(4,6-dimethylpyrimidin-2-yl)-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[4-(2-chloro-4-fluorophenyl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
N-(3-chloro-4-fluorophenyl)-3-[1-(pyrrolidine-3-carbonyl)piperidin-4-yl]propanamide
8-[4-(benzyloxy)butanoyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
4-fluoro-N-{[4-hydroxy-1-(1H-imidazol-4-ylmethyl)azepan-4-yl]methyl}benzene-1-sulfonamide
N-[4-(2-methoxypyridin-3-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
methyl 4-({2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamido}methyl)benzoate
(2S)-2-methoxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-phenylacetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3-phenylpyrrolidine-2,5-dione
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylate
N-[(4-fluorophenyl)methyl]-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)propanamide
2-(oxan-4-yl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-1H-1,3-benzodiazole