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2-[1-(2,2-dimethylpropyl)-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl]ethan-1-ol
3-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-1-[3-(2-methylphenyl)phenyl]urea
N-[1-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
(2S,4S)-4-[(1-benzylpiperidin-4-yl)amino]-1-[(3-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
3-(4-cyclohexylphenyl)-4-(1H-imidazol-2-yl)-1-methyl-1H-pyrazole
4-({5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-ethyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperidin-4-amine
1-methyl-3-[1-(4-methylpentanoyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(4-ethyl-5-{1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-4-ol
1-(4-ethoxypyrimidin-2-yl)-4-phenylpiperidin-4-ol
1-{4-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)piperidin-2-one
(1-methyl-1H-imidazol-2-yl)[1-(4-methylpyridin-2-yl)piperidin-4-yl]methanol
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-methyl-4-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-({[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(2-methyl-1H-indol-1-yl)ethyl]propanamide
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)naphthalen-2-ol
1-(4-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
2-methyl-4-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-6-propylpyrimidine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]propanamide
4-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)but-3-yn-1-ol
N-cyclopentyl-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
(3ar,6ar)-N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(2-{[3-(hydroxymethyl)morpholin-4-yl]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
1-{2-[methyl({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)amino]ethyl}piperidin-2-one
N-(2-hydroxyethyl)-3-(2-hydroxyphenyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
2-methyl-5-(3-methylphenyl)-4-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]pyrimidine
(4aS,8aR)-6-(5-chlorothiophene-2-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N,N-dimethyl-2-[(1S,5R)-3-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-ol
5-ethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
7-(cyclobutylmethyl)-2-[2-(pyridin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-{1-[(1-ethyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}benzoic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(4-chlorophenyl)-3-(2-methoxyethyl)-5-(methoxymethyl)-1H-1,2,4-triazole
1-(5-chloropyridine-3-carbonyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-amine
2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]pyridin-3-ol
(3S,4S)-1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-methyl-5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-acetyl-8-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(diethylamino)ethyl]-N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
4-benzyl-1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine