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5-(2-methoxyacetamido)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
5-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)-2-methylpyridine
1-(1H-indol-5-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
5-acetyl-6-methyl-3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
N,N-dimethyl-2-{methyl[(2,4,5-trimethylphenyl)methyl]amino}propanamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[methyl(pyridin-2-ylmethyl)amino]acetamide
7-methyl-8-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methoxy}quinoline
7-(2-hydroxyethyl)-2-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-oxo-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
(1S,3R)-3-amino-N-[2-(4-chlorophenyl)ethyl]-N-(pyridin-3-ylmethyl)cyclopentane-1-carboxamide
2-[5-(2,5-difluorophenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-(3-methoxypiperidin-1-yl)-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazine
N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
N,N-dimethyl-3-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2,4-dimethylphenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-(2,6-dimethylpyridin-4-yl)-4-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperazine
N-(oxolan-2-ylmethyl)-3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
4-{3-cyclopropyl-5-[2-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-1,2,4-triazol-1-yl}-2-methylpyridine
2-ethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidine-5-carboxamide
(4aS,7aR)-1-(1H-pyrazole-3-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(2,2,2-trifluoro-1-phenylethoxy)ethan-1-one
5-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2E)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-(thiophen-2-yl)prop-2-enamide
1-(cyclopropylmethyl)-4-[(3,4-dimethoxypyridin-2-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
3-{[4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)morpholin-3-yl]-1-(thiomorpholin-4-yl)ethan-1-one
8-[2-(ethylamino)pyrimidine-5-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,6R)-3-(2-propylpyridine-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
7-[(2-fluorophenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-4-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}pyridine-3-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
3-{imidazo[1,2-a]pyridin-3-ylmethyl}-3H,4H-pyrido[4,3-d]pyrimidin-4-one
3-methyl-N-[3-(2-phenylacetamido)phenyl]-1H-pyrazole-5-carboxamide
2-{2-[1-(5-phenylpentanoyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
2-{3-cyclopropyl-5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
1-[2-(2H-1,3-benzodioxol-5-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-benzyl-5-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
4-[4-(3-fluorophenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-8-fluoroquinoline-2-carboxamide
4-(1H-pyrazol-4-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]butan-1-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-methylphenyl)acetamide
N-[(3R,4S)-1-(2-amino-6-methoxypyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide
7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
3-benzyl-4-(2-methanesulfonylacetyl)piperazin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
4-chloro-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrrole-2-carboxamide