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[1-(1-benzothiophen-3-ylmethyl)piperidin-2-yl]methanol
2-({5-[2-amino-3-cyano-6-(4-methylthiophen-2-yl)pyridin-4-yl]pyrimidin-2-yl}amino)acetic acid
4-[(2-methylpyridin-3-yl)oxy]-N-[2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
1-cyclopropyl-N-{3-[methyl(phenyl)amino]propyl}-1H-pyrrole-2-carboxamide
4-[2-(3-methoxyphenoxy)ethyl]-N-(3-methoxyphenyl)piperazine-1-carboxamide
N-{[4-methoxy-3-(pyridin-3-ylmethoxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]cyclohexanecarboxamide
9-(2-methyloxolane-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-1H-indole-3-carboxamide
2-methoxy-5-oxo-6-[3-(pyridin-4-yl)propyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-ethoxy-N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]acetamide
1-{4-methyl-2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-5-yl}ethan-1-one
1-[2-(dimethylamino)ethyl]-4-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-{5-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-[1-(6-cyanopyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
4-{1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-3-yl}benzoic acid
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
(4aS,8aR)-1-(3-aminopropyl)-6-(3-chlorobenzoyl)-decahydro-1,6-naphthyridin-2-one
methyl 4-({5-[(quinolin-8-yloxy)methyl]-1,2-oxazol-3-yl}formamido)butanoate
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-phenylbutan-1-one
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
1-{2,7-diazaspiro[4.5]decan-2-yl}-3-(3-methoxy-4-methylphenyl)propan-1-one
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)quinoxaline-5-carboxamide
(3aR,6aR)-2-cyclopentyl-5-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4S)-4-amino-1-[(2,6-dimethoxyphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
2-(2,4-dichlorophenoxy)-N-(furan-3-ylmethyl)acetamide
1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-cyclohexyl-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
1-methyl-8-[2-(naphthalen-1-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(1-ethynylcyclohexyl)-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
N-[4-(1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1H-imidazol-2-yl)phenyl]acetamide
3-(4-benzoylpiperidin-1-yl)-5-(2,6-dimethoxyphenyl)-1,2,4-triazine
3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
3-[({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}oxy)methyl]pyridine
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-(phenylamino)pyrimidine-5-carboxamide
N-methyl-3-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
2-{5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl}pyridine
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-(1-benzyl-4-hydroxypiperidin-4-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
1-[2-(5-aminopyridin-3-yl)pyrimidin-4-yl]piperidin-4-ol
1-[1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-2-ol
4-ethyl-3-[(1-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3,5,7-trimethyl-2-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-indole
5-(4-fluorophenyl)-N-[2-(1H-indol-1-yl)ethyl]-1,2,4-triazin-3-amine
2-(3-fluorophenoxymethyl)-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide