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4-{5-cyclopropyl-4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-(dimethylamino)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,4-dimethylpyrimidine-5-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(4-methylthiophen-2-yl)pyridine-3-carbonitrile
3-[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(3-{1,4-diazabicyclo[3.2.2]nonan-4-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
3-[1-(2,4-difluoro-3-methoxybenzoyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-1-(1-benzofuran-2-ylmethyl)-4-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]pyrrolidin-3-ol
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-methoxypyrimidin-4-amine
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(2-methylpropyl)pyridin-2-amine
methyl 4-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}benzoate
3-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-methylbut-2-enamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]ethan-1-one
(4aS,8aR)-6-(2-cyclopropylpyrimidine-5-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-3-carboxamide
4-{3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butyl}phenol
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-(benzyloxy)-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-{[3-(4-tert-butylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1S,6R)-3-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-{[6-(5-methyl-1H-indol-3-yl)pyridin-3-yl]methyl}acetamide
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-ethyl-N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
4-[4-(3-methylphenyl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-(6-methoxypyrimidin-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
N-[2-(4-chlorophenyl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-tert-butyl-4-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}furan-2-carboxamide
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-[5-(methoxymethyl)furan-2-carbonyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{3-oxo-9-[4-(1H-pyrazol-4-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
2-({2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(4aS,7aR)-1-(4-chloro-2-hydroxybenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-methyl-N-{[2-(trifluoromethoxy)phenyl]methyl}azepane-2-carboxamide
1-{2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-fluorophenyl)-N-methyl-1,2,4-triazin-3-amine
(2S,4R)-4-amino-1-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
2-[3-(phenoxymethyl)-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazol-1-yl]acetic acid
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
(2E)-N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(2-chlorophenyl)prop-2-enamide
1-[(2,5-dimethylphenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
N-phenyl-N-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}propanamide
2-[(3-{ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}phenyl)amino]acetic acid
[(3R,4R)-1-(4-chloro-1H-pyrazole-3-carbonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol