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({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)[(6-fluoroquinolin-2-yl)methyl]methylamine
3-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridine
2-[4-(2,2-diphenylethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
(3S,4R)-1-cyclobutanecarbonyl-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-(3-chloro-2-methylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
(8R,9aS)-2-(2H-1,3-benzodioxol-5-ylmethyl)-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-(2,4-dimethoxyphenyl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-N-methylpyridin-2-amine
1-(furan-2-ylmethyl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
3-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-6-methoxy-1H-indazole
2-oxo-3-(pentan-3-yl)-1-[3-(pyridin-3-yl)propyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(3aS,6aS)-2-(dimethylcarbamoyl)-5-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-3-yl]propanoic acid
4-({1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperazin-2-one
3-{[5-(1H-imidazol-2-yl)furan-2-yl]sulfanyl}-4-methyl-4H-1,2,4-triazole
methyl 3-(2-methylbutanamido)-5-[(3-methylbutyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{2-[4-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
1-methyl-4-{5-[(2-methyl-1H-imidazol-1-yl)methyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}piperidine
4-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
(2R,3S,6R)-3-(2-methoxyphenyl)-5-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(pyridin-3-yl)-5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]pyrimidine
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
4-hydroxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-({2-[methyl(3-phenylpropyl)carbamoyl]phenyl}amino)acetic acid
1-[1-(3-carbamoylpropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(furan-2-ylmethyl)(3-methylbutan-2-yl)amine
4-[4-(4-cyclohexylpiperazine-1-carbonyl)piperidin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-cyclohexyl-2-(ethylamino)-N-[(4-fluorophenyl)methyl]pyrimidine-5-carboxamide
2-methyl-8-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
3-hydroxy-S-[2-(4-methyl-1,3-thiazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]butane-1-sulfonamido
2-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}-1,3-benzothiazole
1-(oxane-4-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
3-{[4-(3-fluorophenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
5-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-methyl-3-[3-({[(3-propyl-1,2-oxazol-5-yl)methyl]carbamoyl}amino)phenyl]propanamide
N-(1-benzothiophen-2-ylmethyl)-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-(5-acetylthiophen-3-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
3-[(benzenesulfonyl)methyl]-5-[(1R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-1,2,4-oxadiazole
3-(1-benzofuran-2-ylmethyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-methoxypyrimidine-5-carboxamide
1-(pyrrolidin-1-yl)-2-(4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}phenoxy)ethan-1-one
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,3-dimethoxybenzamide
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
2-methoxy-4-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]quinoline
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
4-(1,3-benzothiazol-2-yl)-2-[(2-methylpiperidin-1-yl)methyl]phenol
7-fluoro-4-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]quinazoline