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4-{[3-(4-fluorophenoxy)azetidin-1-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
N-tert-butyl-7-chloro-3,5-dimethyl-1-benzofuran-2-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N,N-dimethyl-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
N-[(2,4-difluorophenyl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-[2-(4-phenylpiperidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-cyclooctyl-5-(4-ethylpiperazine-1-carbonyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methoxyethyl)-N-methylpyridin-2-amine
methyl (2S,4S,5R)-5-(4-chlorophenyl)-4-(cyclobutylcarbamoyl)-1,2-dimethylpyrrolidine-2-carboxylate
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-4-(5-methylfuran-2-yl)benzamide
5-chloro-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-sulfonamide
5-(oxolan-2-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]thiophene-2-carboxamide
2-(methylsulfanyl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}cyclohexanecarboxamide
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(naphthalen-1-yl)ethan-1-one
(1S,5R)-6-benzyl-3-[(3-ethoxy-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-2-[(1S,5R)-6-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4'-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[({1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]-N-methylacetamide
2-{4-[(3,5-difluorophenyl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(1H-imidazol-1-yl)ethyl]-3-[(2-phenylethyl)amino]-5-(pyrrolidine-1-sulfonyl)benzamide
N-(3-chloro-2-methylphenyl)-3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-3-oxopropanamide
(2S,4S)-4-amino-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
(3R,4R)-3-cyclopropyl-1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-methylpyrrolidin-3-ol
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
6-methyl-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
ethyl 1-[2-(methylsulfanyl)pyridine-3-carbonyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
6-ethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-N-(3-methoxypropyl)benzene-1-sulfonamide
5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-indole
1-[2-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
2-ethoxy-5-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
5-(methoxymethyl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
3-[2-(azetidin-1-yl)-2-oxoethyl]-1-[(2-fluorophenyl)methyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)acetamide
N-(3,5-dimethoxyphenyl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)propanamide
1-[3-(2,3-dihydro-1-benzofuran-5-yl)benzoyl]pyrrolidine
1-[2-(1H-imidazol-2-yl)ethyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-(2-hydroxypropanoyl)piperidine-4-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(4-methylphenyl)propanoyl]piperidin-3-yl}propanamide
methyl 2-[3-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)-1H-indol-1-yl]acetate
N-[2-ethyl-4-(3-methyl-1H-pyrazol-1-yl)phenyl]acetamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-3-carboxamide
(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol