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[1-(2-fluorophenyl)propan-2-yl]({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl})amine
6-(2-chlorophenyl)-2-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-(4-chlorophenyl)-1-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)butan-1-one
1-[2-butyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]pentane-1,2-dione
(3R,4R)-4-amino-1-({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)piperidin-3-ol
[3-(cyclopropylmethyl)-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl]methanol
2-(4-{4-[4-(pyridin-4-yl)piperidin-1-yl]piperidin-1-yl}benzoyl)-1,2,3,4-tetrahydroisoquinoline
[(2S,6S)-4-{imidazo[1,2-a]pyridin-2-ylmethyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[(3S)-3-ethylmorpholin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-cyclopropyl-3-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
4-{2-oxo-2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
[(3S,5R)-1-(5-chloro-2-fluorobenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
8-(hex-5-en-1-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[7-(2-methoxy-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,6,8-trimethylquinoline-4-carboxamide
4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-6-fluoro-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-({2-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(1H-pyrazol-1-ylmethyl)piperidine
(1R,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2,5-dimethylphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-[1-(furan-3-ylmethyl)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-yl]ethan-1-ol
2-(dimethylamino)-2-(3-fluorophenyl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
2,5-dimethyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrazine
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(1S,5R)-3-(oxan-4-yl)-6-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
3-{5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}benzonitrile
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
(2S)-2-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-phenylacetamide
2-chloro-N-{2-[3-(methylsulfanyl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
1-(4-phenyl-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethan-1-one
7-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2R,4S)-4-hydroxy-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidine-2-carboxylic acid
2-(dimethylamino)-2-(3-methylphenyl)-1-[3-(morpholin-4-yl)azetidin-1-yl]ethan-1-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-cyclopentyl-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
3-cyclopropyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-{2-[4-(methylsulfanyl)phenyl]acetyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2-methyl-1H-pyrrole-3-carbonyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-methyl-N-(3-methylbutyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3aR,6aR)-2-benzyl-N-(furan-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})[(3-methylpyridin-4-yl)methyl]amine
(1S,5R)-6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(4-fluorophenyl)ethyl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N,N,1-triethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-methyl-2-phenylpiperazine-1-carboxamide
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propanamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide