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(3R,4S)-4-cyclopropyl-1-(3-methoxy-2-methylbenzoyl)pyrrolidin-3-amine
N-[(3R,4R)-3-hydroxy-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl]pyridine-4-carboxamide
3-{5-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
3-[(3R,4S)-4-(dimethylamino)-1-[2-(dimethylamino)benzoyl]piperidin-3-yl]propan-1-ol
N-{[2-(dimethylamino)pyridin-3-yl]methyl}quinoline-8-carboxamide
5-hydroxy-2-(4-methylphenyl)-6-[2-(trifluoromethyl)morpholine-4-carbonyl]-2,3-dihydropyridazin-3-one
1-{1-[6-(propan-2-yl)-1H-indole-2-carbonyl]piperidin-3-yl}pyrrolidin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 2,4-dimethyl-5-[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})carbamoyl]-1H-pyrrole-3-carboxylate
[(1-ethylpiperidin-3-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
[1-(2-fluorophenyl)propan-2-yl]({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl})amine
5-oxo-1-{[1-(piperidin-1-yl)cyclopentyl]methyl}pyrrolidine-3-carboxylic acid
2-(but-3-enoyl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-chloro-2-fluorophenyl)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)urea
3-chloro-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
methyl 5-[2-(1,2,3,6-tetrahydropyridin-4-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1-[4-(4-methoxyphenoxy)phenyl]urea
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-[2-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
N-(pyridin-3-ylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-methanesulfonyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyrrolidine-2-carboxamide
(3R,4R)-1-(2-methoxyquinoline-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-{[(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-(2-ethoxyethyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
2-(1-{[1-(furan-3-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
methyl N-{2-[4-(1H-indazol-5-yl)-3-oxopiperazin-1-yl]-2-oxoethyl}carbamate
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,3-difluoropiperidine
3-[1-(3-chlorophenyl)cyclopropyl]-1-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-[(2-methoxyphenyl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)pyrazine-2-carboxamide
1-[1-(2-methylpropanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(2-phenylpropyl)(pyridin-4-ylmethyl)amine
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-one
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]oxolane-2-carboxamide
(1R,5R)-6-{[2-(methylsulfanyl)phenyl]methyl}-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(benzyloxy)ethyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
2-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}quinolin-8-ol
8-cyclopropanecarbonyl-2-(3-phenylpropanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(1H-imidazol-2-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-benzyl-N-ethyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
4-({[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
5-cyclopropanecarbonyl-1'-(1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
9-(4-hydroxybenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenylethan-1-one
5-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-1-ethyl-1H-pyrazole-4-sulfonamide