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N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
2-amino-1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
2-{4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
2-(dimethyl-1,3-thiazol-5-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]acetamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-(2-tert-butylphenyl)-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
2-(morpholine-4-carbonyl)-N-[4-(pyridin-2-yl)butyl]pyridin-4-amine
8-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
8-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2,3-dihydro-1-benzofuran-7-carbonyl)-2-(trifluoromethyl)morpholine
3,5-dimethyl-N-[3-(methylsulfanyl)propyl]-1-benzofuran-2-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-[(thiolan-3-yl)amino]pyridine-3-carboxamide
2-(4-fluorophenyl)-1-{4-[3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}ethan-1-one
4-(5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}furan-2-yl)-2-methylbut-3-yn-2-ol
methyl (2S)-2-(2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetamido)-2-phenylacetate
3-({[2-(dimethylamino)ethyl][(3-methylthiophen-2-yl)methyl]amino}methyl)-N-methylpyridin-2-amine
N-{2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]thiophen-3-yl}acetamide
4-methyl-2-(2-propyl-1H-imidazol-1-yl)pyridine
(3S,4S)-1-(6-methylpyridazin-3-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)spiro[azepane-4,2'-chromene]
2-(ethylamino)-N-methyl-N-(quinolin-8-ylmethyl)pyrimidine-5-carboxamide
[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl](pentan-3-yl)amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(thiophen-3-yl)ethan-1-one
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methylpyrimidin-2-amine
N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2-(pyrrolidin-3-yl)benzamide
N,8-dimethyl-3-(morpholin-4-ylmethyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-2-one
5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]thiophene-2-carboxamide
1-(2-fluorophenyl)-4-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]piperazine
2,7-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
2-ethyl-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-phenoxyethan-1-one
3-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}benzonitrile
2-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(pyrrolidin-1-yl)ethan-1-one
2-benzyl-N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1,3-benzoxazole-5-carboxamide
3-fluoro-2-(2,3,4-trimethoxyphenyl)pyridine
3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
2-(2-phenylethyl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,3-benzoxazole
4-[2-(4-methoxyphenyl)ethyl]-11-(1,2,3,4-tetrahydroisoquinolin-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(4-{2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-3-(1,2-oxazolidin-2-yl)propanamide
(2S,4R)-1-[(2-hydroxy-4-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-4-(thian-4-yl)piperazine
N-[2-(3-chlorophenyl)ethyl]-1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
4-ethyl-3-(1-ethyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(dimethylsulfamoyl)ethyl]-5-methyl-1H-indazole-3-carboxamide
4-(3-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)-2-methylbutan-2-ol