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1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(3R,4R)-4-cyclopropyl-3-methyl-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-ol
2-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(4-methylphenyl)quinoline-4-carbonyl]-1,2-oxazolidin-4-ol
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N,1,3-trimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(5-chloro-2-methylphenyl)piperazine
1-[2-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}phenoxy)ethyl]-3-methylpiperidine
5-(4-cyclohexanecarbonylpiperazine-1-carbonyl)-2-ethylpyrimidine
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(oxolan-2-ylmethyl)piperidin-4-amine
N-ethyl-7-{[3-(1H-imidazol-1-yl)propyl]sulfamoyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-{[(2,6-difluorophenyl)methyl]carbamoyl}-5-methoxybenzoic acid
(4aS,7aR)-1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-fluoro-4-methoxyphenyl)-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-1,2,3-triazole
2-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-N-[(2-methylphenyl)methyl]acetamide
1-[5-(1H-1,3-benzodiazol-2-ylmethyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
5-methoxy-3-[(2R)-pyrrolidin-2-ylmethyl]-3,4-dihydroquinazolin-4-one
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1,1-dioxo-1λ6-thiolane-3-carboxamide
N1-(4-methylpyridin-2-yl)-N2-[4-(propan-2-yl)pyrimidin-2-yl]ethane-1,2-diamine
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylacetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[({1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}amino)methyl]phenol
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
5-(1H-indol-4-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
(3S,4R)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-4-methylpiperidine-3,4-diol
2,2-dimethyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
4-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
5-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,3,4-oxadiazol-2-amine
2-(4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
methyl 2-(2-chloro-4,5-dimethoxyphenyl)-1H-1,3-benzodiazole-6-carboxylate
(1R,3S)-3-ethoxy-7-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
(2R,3S,6R)-5-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-(cyclohexylmethyl)-2-(propane-1-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}piperidin-2-one
2-(4-fluoro-2-methoxyphenyl)-5-(1H-imidazol-1-ylmethyl)pyridine
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]methylamine
6-(furan-3-yl)-4-methyl-1,2-dihydroquinolin-2-one
3-(2-{[2-(2-aminoethyl)quinazolin-4-yl]amino}ethyl)-1,3-oxazinan-2-one
(4-{[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}oxan-4-yl)methanol
N,4-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-phenyl-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
5-(1-benzylpiperidin-4-yl)-3-cyclopentyl-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
4-{1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}-1,4-oxazepan-6-ol
(3aS,7aR)-5-methyl-2-(1-methyl-1H-pyrrole-2-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3S,9aR)-3-methyl-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,2,3,3-tetramethyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]cyclopropane-1-carboxamide