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3,3-dimethyl-1-[(5-{[4-(propan-2-yloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
1-{4-[(dicyclopropylmethyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-({1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]pyrrolidin-3-yl}methyl)benzamide
N-tert-butyl-2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1R,4S)-N,1,7,7-tetramethyl-3-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-oxabicyclo[2.2.1]heptane-4-carboxamide
5-(azepane-1-carbonyl)-N-benzyl-N-methyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{3-[4-({[(3-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(benzylsulfamoyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
methyl N-[1-({[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}carbamoyl)ethyl]carbamate
4-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]benzoic acid
5-(3,3-diphenylpiperidine-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
1-(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,4-diazepan-5-one
N-[2-methyl-2-(morpholin-4-yl)propyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
8-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-yl]methanol
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2,5-trimethylfuran-3-carboxamide
8-(1-hydroxypropan-2-yl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(1H-pyrrol-1-yl)pentanoyl]piperidine-4-carboxylic acid
4-(3-amino-1H-indazol-5-yl)-N,N-dimethylbenzamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}acetamide
N-benzyl-N-ethyl-2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-hydroxyethan-1-one
(4S)-1-(3-hydroxy-1,2-oxazole-5-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
methyl({2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}){[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}amine
4-fluorophenyl (7S,9aR)-7-[(4-chlorophenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
[(3R,4S)-1-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
3-(diethylamino)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
N-[(3S,4R)-1-[1-(2-fluorophenyl)piperidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-cyclopropyl-5-[4-(4-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
4-{[1-(3-methoxyphenyl)propan-2-yl]amino}-N-phenylpiperidine-1-carboxamide
ethyl 3-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)amino]propanoate
3-(2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
3-methyl-8-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
2-ethyl-8-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-chloro-3-({[2-(2,6-dimethylphenoxy)ethyl](ethyl)amino}methyl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
8-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
5-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrimidine
2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
4-phenoxy-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylic acid
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-(propan-2-yloxy)benzamide
1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
{2-oxo-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethyl}urea