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N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-{[2-({[6-(methoxymethyl)pyrimidin-4-yl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
1-(4-fluorophenyl)-4-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
N-methyl-4-{[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]methyl}benzamide
2-[benzyl({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]ethan-1-ol
N-(butan-2-yl)-4-methanesulfonyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1,1,1-trifluoro-3-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-2-ol
3-butyl-4-(4-hydroxy-2-methylpyrimidine-5-carbonyl)-1-methylpiperazin-2-one
[(1R,3S,3aS,6aR)-1-ethyl-5-methyl-3-(3-phenoxyphenyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-(1,2-oxazol-3-ylmethyl)urea
2-ethoxy-5-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]pyridine
(2S,4R)-1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
2-methoxy-3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrazine
9-ethyl-4-(4-fluorobenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(5-aminopyridin-3-yl)-N,N,5,6-tetramethylpyrimidin-2-amine
3-[(3R,4S)-1-(3-fluoro-4-methoxybenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(3S,4S)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-propylpyrrolidine-3-carboxylic acid
3-(4-chloro-1H-pyrazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
2,6-dimethyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]quinoline-4-carboxamide
2-[5-(2H-1,3-benzodioxol-5-yl)-1-cyclohexyl-1H-1,2,4-triazol-3-yl]acetamide
3-fluoro-4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
1-(2-methylfuran-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]amine
3-[2-(dimethylamino)ethyl]-1-ethyl-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(3R,4S)-3-[(2-aminopyrimidin-4-yl)amino]-4-cyclopropylpyrrolidine-1-carbonyl]oxane-4-carbonitrile
4-[2-(adamantan-1-yl)acetyl]-3-benzylpiperazin-2-one
N-(oxan-4-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
7-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-4H-chromen-4-one
2-amino-3-ethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-methyl-9-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
4-(cyclopropylmethyl)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
3-[(3-methylquinoxalin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methoxy-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
8-[(5-carboxyfuran-2-yl)methyl]-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2,3-difluorophenoxymethyl)-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-1,3-oxazole-4-carboxamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-[methyl(1,3-thiazol-2-ylmethyl)amino]azepan-2-one
methyl 5-[(1-methylpiperidin-4-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-4-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
2-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](furan-2-ylmethyl)amino}butan-1-ol
3-({3-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}(methyl)amino)-1λ6-thiolane-1,1-dione
1-[2-methoxy-4-(thiomorpholin-4-ylmethyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2,2-dimethyloxane-4-carboxamide
2-(diethylamino)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylacetamide
3-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}phenol
(4aR,8aR)-2-methanesulfonyl-7-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide