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3-hydroxy-S-(2-pentanoyl-1,2,3,4-tetrahydroisoquinolin-6-yl)butane-1-sulfonamido
4-[3-(ethoxymethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-1-oxaspiro[4.5]decan-2-one
2-chloro-5-acetamido-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
4-[(diethylamino)methyl]-N,5-diethyl-N-[(1R,2R)-2-hydroxycyclohexyl]furan-2-carboxamide
2-{[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-4-methoxypyridine
ethyl({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-ethyl-7-methoxy-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]imidazo[1,2-a]pyridine-6-carboxamide
3-{[1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{[6-({[2-(dimethylamino)pyridin-3-yl]methyl}amino)pyrimidin-4-yl]amino}ethan-1-ol
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
6-[(2S)-1-cyclohexyl-3-hydroxypropan-2-yl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
2-(2-fluorophenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{[1-(1H-indol-2-ylmethyl)piperidin-3-yl]methyl}-2-methoxyacetamide
2-amino-4-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-benzothiazole-6-carboxamide
2-({2-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
N-{2-methyl-1-[7-(3-methylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}oxolane-3-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
N-cyclopropyl-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
4-phenyl-N-(1-propyl-1H-1,2,4-triazol-3-yl)azepane-1-carboxamide
[(1-methyl-1H-imidazol-2-yl)methyl]({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
1-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-4-yl]piperidin-4-ol
7-acetamido-N-[(2-fluorophenyl)methyl]-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-ethyl-3-(3-fluoro-4-methylphenyl)-6-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
ethyl 1-[(4-acetamidophenyl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
(2R,3S,6R)-5-(furan-3-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
3-(3-methoxypropyl)-1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidine-3-carboxylic acid
N-cyclopropyl-N-(1-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
3-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-[2-(1,3,4-oxadiazol-2-yl)phenyl]urea
2-[(2,6-dichlorophenyl)methyl]-5-(morpholine-4-carbonyl)pyrimidin-4-ol
2-(3-methoxypropyl)-8-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-({[(3-{2-[4-(4-hydroxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
N-(1-oxo-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-2-yl)methanesulfonamide
2-(hydroxymethyl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 3-{[4-(4-methoxyphenoxy)phenyl]formamido}propanoate
2-{2-[1-(4-chloro-2-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-[1-(methoxymethyl)cyclobutanecarbonyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-({1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-3-yl}methyl)pyridine-2-carboxamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-4-hydroxy-2-methylpyrimidine-5-carboxamide