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N2,N2-dimethyl-6-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyrimidine-2,4-diamine
3-[(4aR,7aS)-4-[(2-ethoxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-cyclopentanecarbonyl-N-methyl-N-(1H-pyrazol-3-ylmethyl)piperidine-4-carboxamide
3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[3-(pyridin-4-yl)propyl]propanamide
2-chloro-4-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1H-pyrazole
4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]-N-(2-phenylphenyl)piperidine-1-carboxamide
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-2-fluorobenzamide
N-(3-chloro-4-methoxyphenyl)-6-(3-methylbutyl)-6-azaspiro[2.5]octane-1-carboxamide
2-(2,4-difluorophenyl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methylpyrazine
N-[4-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]acetamide
3-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1-(thiophen-2-yl)urea
1-{[5-(3-cyclohexyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpiperazine
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)furan-3-carboxamide
(4aS,8aS)-2-(3-phenoxybenzoyl)-decahydro-2,7-naphthyridin-4a-ol
8-fluoro-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
4-benzyl-1-[(3,4-dimethoxypyridin-2-yl)methyl]pyrrolidin-2-one
2-{1-cyclohexyl-4-[1-(3-methoxyphenyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-ethyl-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(2R)-2-amino-3-(furan-2-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
2-(2,3,4-trimethoxyphenyl)benzamide
2-methyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-3,4-dihydropyrimidin-4-one
N-{[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]methyl}-4-phenylbenzamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
N-(isoquinolin-5-ylmethyl)-N-methyl-N'-[2-(methylsulfanyl)phenyl]butanediamide
(3aS,6aS)-2-methyl-5-[2-(4-phenylphenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-4-(hydroxymethyl)-1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-3-ol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidine
N-[4-(3-methylphenyl)phenyl]-1-[(2R)-oxolane-2-carbonyl]piperidine-4-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}acetamide
N-(3-methoxypropyl)-1-methyl-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(3,4,5-trifluorophenyl)ethan-1-one
2-(5-tert-butyl-2H-1,2,3,4-tetrazol-2-yl)-N-(1-cyclohexyl-1H-pyrazol-5-yl)acetamide
6-(2-chlorophenyl)-7-methyl-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine
(2S,4S)-4-cyclobutaneamido-N,1-dimethyl-N-(quinolin-8-ylmethyl)pyrrolidine-2-carboxamide
7-(cyclopropylmethyl)-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decane
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[(2-methylphenyl)sulfanyl]piperidine
1-(4-{4-[2-(2-hydroxyethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)-3-methoxypropan-1-one
(2S,4R)-N-methyl-4-{[(3-phenoxyphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
methyl (2S,4S)-1-{[4-(propan-2-yl)phenyl]methyl}-4-(pyridine-2-amido)pyrrolidine-2-carboxylate
1-(4-methylquinazolin-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}pyrrolidine-2-carboxamide
3-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-[1-(oxan-4-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N4-[(5-methylpyrazin-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(aminomethyl)-N-(2-fluoro-5-methylphenyl)piperidine-1-carboxamide